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1 . Academic Journal
How to identify and eliminate compounds with a risk of high clinical dose during the early phase of lead optimisation in drug discovery
저자
by
Teague, Simon
;
Valko, Klara
.
소스
In
European Journal of Pharmaceutical Sciences
15 December 2017 110:37-50
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4 . Academic Journal
iBCS: 3. A Biopharmaceutics Classification System for Orally Inhaled Drug Products.
저자
by
Hastedt, Jayne E.
;
Bäckman, Per
;
Cabal, Antonio
;
Clark, Andy
;
Ehrhardt, Carsten
, et al.
소스
Molecular Pharmaceutics; 1/1/2024, Vol. 21 Issue 1, p164-172, 9p
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7 . Academic Journal
iBCS: 1. Principles and Framework of an Inhalation-Based Biopharmaceutics Classification System.
저자
by
Hastedt, Jayne E.
;
Bäckman, Per
;
Cabal, Antonio
;
Clark, Andy
;
Ehrhardt, Carsten
, et al.
소스
Molecular Pharmaceutics; 7/4/2022, Vol. 19 Issue 4, p2032-2039, 8p
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7 . Periodical
Investigation of Janus Kinase (JAK) Inhibitors for Lung Delivery and the Importance of Aldehyde Oxidase Metabolism
저자
by
Wellaway, Christopher R.
;
Baldwin, Ian R.
;
Bamborough, Paul
;
Barker, Daniel
;
Bartholomew, Michelle A.
, et al.
소스
Journal of Medicinal Chemistry; January 2022, Vol. 65 Issue: 1 p633-664, 32p
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7 . Academic Journal
Multimodal imaging of drug and excipients in rat lungs following an inhaled administration of controlled-release drug laden PLGA microparticles.
저자
by
Robinson, Eve
;
Giffen, Paul
;
Hassall, Dave
;
Ball, Doug
;
Reid, Heather
, et al.
소스
Analyst
. 5/21/2021, Vol. 146 Issue 10, p3378-3390. 13p.
Full Text (RSC Gold)
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7 . Academic Journal
Substituted indole-1-acetic acids as potent and selective CRTh2 antagonists—discovery of AZD1981
저자
by
Luker, Tim
;
Bonnert, Roger
;
Brough, Steve
;
Cook, Anthony R.
;
Dickinson, Mark R.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(21):6288-6292
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7 . Academic Journal
Acylglycinamides as inhibitors of glycine transporter type 1
저자
by
Blunt, Richard
;
Porter, Roderick
;
Johns, Amanda
;
Nash, David
;
Puckey, Gemma
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(20):6176-6179
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7 . Academic Journal
Identification of novel α7 nAChR positive allosteric modulators with the use of pharmacophore in silico screening methods
저자
by
Capelli, Anna Maria
;
Castelletti, Laura
;
Salvagno, Cristian
;
Oliosi, Beatrice
;
Di Lenarda, Elisa
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 August 2010 20(15):4561-4565
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7 . Academic Journal
Structure-driven HtL: Design and synthesis of novel aminoindazole inhibitors of c-Jun N-terminal kinase activity
저자
by
Stocks, Michael J.
;
Barber, Simon
;
Ford, Rhonan
;
Leroux, Frederic
;
St-Gallay, Steve
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2005 15(14):3459-3462
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7 . Periodical
iBCS: 3. A Biopharmaceutics Classification System for Orally Inhaled Drug Products
저자
by
Hastedt, Jayne E.
;
Bäckman, Per
;
Cabal, Antonio
;
Clark, Andy
;
Ehrhardt, Carsten
, et al.
소스
Molecular Pharmaceutics; 20230101, Issue: Preprints
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