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1 . Academic Journal
A TRIM21-based bioPROTAC highlights the therapeutic benefit of HuR degradation.
저자
by
Fletcher, Alice
;
Clift, Dean
;
de Vries, Emma
;
Martinez Cuesta, Sergio
;
Malcolm, Timothy
, et al.
소스
Nature Communications; 11/4/2023, Vol. 14 Issue 1, p1-14, 14p
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7 . Academic Journal
Targeting a Novel KRAS Binding Site: Application of One-Component Stapling of Small (5–6-mer) Peptides.
저자
by
Fumagalli, Gabriele
;
Carbajo, Rodrigo J.
;
Nissink, J. Willem M.
;
Tart, Jonathan
;
Dou, Rongxuan
, et al.
소스
Journal of Medicinal Chemistry; 12/9/2021, Vol. 64 Issue 23, p17287-17303, 17p
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7 . Periodical
Identification and Characterization of Dual Inhibitors of the USP25/28 Deubiquitinating Enzyme Subfamily
저자
by
Wrigley, Jonathan D.
;
Gavory, Gerald
;
Simpson, Iain
;
Preston, Marian
;
Plant, Helen
, et al.
소스
ACS Chemical Biology; 20240101, Issue: Preprints
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7 . Academic Journal
Rapid Identification of Novel Allosteric PRC2 Inhibitors.
저자
by
Read, Jon A.
;
Tart, Jonathan
;
Rawlins, Philip B.
;
Gregson, Clare
;
Jones, Karen
, et al.
소스
ACS Chemical Biology; Oct2019, Vol. 14 Issue 10, p2134-2140, 7p
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7 . Academic Journal
Small Molecule Binding Sites on the Ras:SOS Complex Can Be Exploited for Inhibition of Ras Activation.
저자
by
Winter, Jon J. G.
;
Anderson, Malcolm
;
Blades, Kevin
;
Brassington, Claire
;
Breeze, Alexander L.
, et al.
소스
Journal of Medicinal Chemistry
. Mar2015, Vol. 58 Issue 5, p2265-2274. 10p.
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7 . Academic Journal
Matrix metalloproteinase 17 is necessary for cartilage aggrecan degradation in an inflammatory environment
저자
by
Clements, Kristen M
;
Flannelly, Jo K
;
Tart, Jonathan
;
Brockbank, Sarah M V
;
Wardale, John
, et al.
소스
Annals of Rheumatic Diseases
. Apr 01, 2011 70(4):683-689
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7 . Academic Journal
Design and Synthesis of Novel Lactate Dehydrogenase A Inhibitors by Fragment-Based Lead Generation.
저자
by
Ward, Richard A.
;
Brassington, Claire
;
Breeze, Alexander L.
;
Caputo, Alessandro
;
Critchlow, Susan
, et al.
소스
Journal of Medicinal Chemistry
. 4/12/2012, Vol. 55 Issue 7, p3285-3306. 22p.
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7 . Academic Journal
Integrin α
5
β
1
and ADAM-17 Interact in Vitro and Co-localize in Migrating HeLa Cells.
저자
by
Bax, Daniel V.
;
Messent, Anthea J.
;
Tart, Jonathan
;
van Hoang, Mien
;
Kott, Jan
, et al.
소스
Journal of Biological Chemistry
. 5/24/2004, Vol. 279 Issue 21, p22377-22386. 10p. 24 Color Photographs, 2 Black and White Photographs, 1 Diagram, 10 Graphs.
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7 . Academic Journal
Identification and Characterization of Dual Inhibitors of the USP25/28 Deubiquitinating Enzyme Subfamily
저자
by
Wrigley, Jonathan D.
;
Gavory, Gerald
;
Simpson, Iain
;
Preston, Marian
;
Plant, Helen
, et al.
소스
ACS CHEMICAL BIOLOGY
; DEC 2017, 12 12, p3113-p3125, 13p.
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7 . Periodical
Mutations in the Interglobular Domain of Aggrecan Alter Matrix Metalloproteinase and Aggrecanase Cleavage Patterns
저자
by
Mercuri, Francesca A.
;
Maciewicz, Rose A.
;
Tart, Jonathan
;
Last, Karena
;
Fosang, Amanda J.
.
소스
Journal of Biological Chemistry; October 2000, Vol. 275 Issue: 42 p33038-33045, 8p
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