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1 . Academic Journal
Drug–Drug Interactions Related to Altered Absorption and Plasma Protein Binding: Theoretical and Regulatory Considerations, and an Industry Perspective
저자
by
Hochman, Jerome
;
Tang, Cuyue
;
Prueksaritanont, Thomayant
.
소스
In
Journal of Pharmaceutical Sciences
March 2015 104(3):916-929
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5 . Academic Journal
A dynamic view to the modulation of phosphorylation and O-GlcNAcylation by inhibition of O-GlcNAcase
저자
by
Tang, Cuyue
;
Welty, Devin F.
.
소스
In
Computational Biology and Chemistry
August 2013 45:9-16
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4 . Academic Journal
Identification of second-generation P2X3 antagonists for treatment of pain
저자
by
Ginnetti, Anthony T.
;
Paone, Daniel V.
;
Stauffer, Shaun R.
;
Potteiger, Craig M.
;
Shaw, Anthony W.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 May 2018 28(8):1392-1396
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7 . Academic Journal
Conformational-Design-Driven Discovery of EZM0414: A Selective, Potent SETD2 Inhibitor for Clinical Studies.
저자
by
Alford, Joshua S.
;
Lampe, John W.
;
Brach, Dorothy
;
Chesworth, Richard
;
Cosmopoulos, Kat
, et al.
소스
ACS Medicinal Chemistry Letters; 7/14/2022, Vol. 13 Issue 7, p1137-1143, 7p
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7 . Academic Journal
Simultaneous determination of urinary free cortisol and 6β-hydroxycortisol by liquid chromatography–atmospheric pressure chemical ionization tandem mass spectrometry and its application for estimating hepatic CYP3A induction
저자
by
Tang, Cuyue
;
Kassahun, Kelem
;
McIntosh, Ian S
;
Brunner, Janice
;
Rodrigues, A.David
.
소스
In
Journal of Chromatography B: Biomedical Sciences and Applications
2000 742(2):303-313
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7 . Academic Journal
Discovery of 5-aryl-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-ones as positive allosteric modulators of metabotropic glutamate subtype-2 (mGlu2) receptors with efficacy in a preclinical model of psychosis
저자
by
Layton, Mark E.
;
Reif, Alexander J.
;
Hartingh, Timothy J.
;
Rodzinak, Kevin
;
Dudkin, Vadim
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 February 2016 26(4):1260-1264
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7 . Academic Journal
Discovery of a First-in-Class Inhibitor of the Histone Methyltransferase SETD2 Suitable for Preclinical Studies.
저자
by
Lampe, John W.
;
Alford, Joshua S.
;
Boriak-Sjodin, P. Ann
;
Brach, Dorothy
;
Cosmopoulos, Kat
, et al.
소스
ACS Medicinal Chemistry Letters; 10/14/2021, Vol. 12 Issue 10, p1539-1545, 7p
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7 . Academic Journal
Discovery of the Oxadiazine FRM-024: A Potent CNS-Penetrant Gamma Secretase Modulator.
저자
by
Bursavich, Matthew G.
;
Harrison, Bryce A.
;
Acharya, Raksha
;
Costa, Donald E.
;
Freeman, Emily A.
, et al.
소스
Journal of Medicinal Chemistry; 10/14/2021, Vol. 64 Issue 19, p14426-14447, 22p
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7 . Academic Journal
Discovery of 2,5-diarylnicotinamides as selective orexin-2 receptor antagonists (2-SORAs)
저자
by
Mercer, Swati P.
;
Roecker, Anthony J.
;
Garson, Susan
;
Reiss, Duane R.
;
Meacham Harrell, C.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2013 23(24):6620-6624
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7 . Academic Journal
Identification of a First-in-Class SETD2 Inhibitor That Shows Potent and Selective Anti-Proliferative Activity in t(4;14) Multiple Myeloma: T(4;14) Multiple Myeloma Cells Are Dependent on Both H3K36 Di and Tri-Methylation
저자
by
Thomenius, Michael J
;
Totman, Jennifer
;
Cosmopoulos, Kat
;
Brach, Dorothy
;
Ci, Lei
, et al.
소스
In
Blood
29 November 2018 132 Supplement 1:3207-3207
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