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1 . Academic Journal
Spiro heterocycles bearing piperidine moiety as potential scaffold for antileishmanial activity: synthesis, biological evaluation, and in silico studies
저자
by
Mounir A. A. Mohamed
;
Asmaa M. Kadry
;
Salma A. Bekhit
;
Mohammed A. S. Abourehab
;
Kikuko Amagase
, et al.
소스
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1, Pp 330-342 (2023)
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7 . Academic Journal
Discovery of new pyridine-quinoline hybrids as competitive and non-competitive PIM-1 kinase inhibitors with apoptosis induction and caspase 3/7 activation capabilities
저자
by
Mostafa M. M. El-Miligy
;
Marwa E. Abdelaziz
;
Salwa M. Fahmy
;
Tamer M. Ibrahim
;
Marwa M. Abu-Serie
, et al.
소스
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1 (2023)
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7 . Academic Journal
Using CADD tools to inhibit the overexpressed genes FAP, FN1, and MMP1 by repurposing ginsenoside C and Rg1 as a treatment for oral cancer
저자
by
Manal Abouelwafa
;
Tamer M. Ibrahim
;
Mohamed S. El-Hadidi
;
Mater H. Mahnashi
;
Amani Y. Owaidah
, et al.
소스
Frontiers in Molecular Biosciences, Vol 10 (2023)
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7 . Academic Journal
Structure-guided approach on the role of substitution on amide-linked bipyrazoles and its effect on their anti-inflammatory activity
저자
by
Souraya A. Domiati
;
Khaled H. Abd El Galil
;
Mohammed A. S. Abourehab
;
Tamer M. Ibrahim
;
Hanan M. Ragab
.
소스
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 2179-2190 (2022)
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7 . Academic Journal
New pyrazolylpyrazoline derivatives as dual acting antimalarial-antileishamanial agents: synthesis, biological evaluation and molecular modelling simulations
저자
by
Adnan A. Bekhit
;
Eskedar T. Lodebo
;
Ariaya Hymete
;
Hanan M. Ragab
;
Salma A. Bekhit
, et al.
소스
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 2320-2333 (2022)
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7 . Academic Journal
In silico identification of novel SARS-COV-2 2′-O-methyltransferase (nsp16) inhibitors: structure-based virtual screening, molecular dynamics simulation and MM-PBSA approaches
저자
by
Mahmoud A. El Hassab
;
Tamer M. Ibrahim
;
Sara T. Al-Rashood
;
Amal Alharbi
;
Razan O. Eskandrani
, et al.
소스
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 36, Iss 1, Pp 727-736 (2021)
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7 . Academic Journal
In Silico Targeting of Fascin Protein for Cancer Therapy: Benchmarking, Virtual Screening and Molecular Dynamics Approaches
저자
by
Heba H. A. Hassan
;
Muhammad I. Ismail
;
Mohammed A. S. Abourehab
;
Frank M. Boeckler
;
Tamer M. Ibrahim
, et al.
소스
Molecules, Vol 28, Iss 3, p 1296 (2023)
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7 . Academic Journal
Design and synthesis of phthalazine-based compounds as potent anticancer agents with potential antiangiogenic activity via VEGFR-2 inhibition
저자
by
Salwa Elmeligie
;
Asmaa M. Aboul-Magd
;
Deena S. Lasheen
;
Tamer M. Ibrahim
;
Tamer M. Abdelghany
, et al.
소스
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 34, Iss 1, Pp 1347-1367 (2019)
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7 . Academic Journal
Supporting SARS-CoV-2 Papain-Like Protease Drug Discovery: In silico Methods and Benchmarking
저자
by
Tamer M. Ibrahim
;
Muhammad I. Ismail
;
Matthias R. Bauer
;
Adnan A. Bekhit
;
Frank M. Boeckler
.
소스
Frontiers in Chemistry, Vol 8 (2020)
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7 . Academic Journal
Development of Novel Quinoline-Based Sulfonamides as Selective Cancer-Associated Carbonic Anhydrase Isoform IX Inhibitors
저자
by
Moataz Shaldam
;
Alessio Nocentini
;
Zainab M. Elsayed
;
Tamer M. Ibrahim
;
Rofaida Salem
, et al.
소스
International Journal of Molecular Sciences, Vol 22, Iss 20, p 11119 (2021)
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