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1 . Academic Journal
Design, synthesis, and biological evaluation of phenylcyclopropylamine-entinostat conjugates that selectively target cancer cells
저자
by
Ota, Yosuke
;
Itoh, Yukihiro
;
Takada, Yuri
;
Yamashita, Yasunobu
;
Hu, Chenliang
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 February 2024 100
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7 . Academic Journal
Structural optimization of a lysine demethylase 5 inhibitor for improvement of its cellular activity
저자
by
Terao, Mitsuhiro
;
Yamashita, Yasunobu
;
Takada, Yuri
;
Itoh, Yukihiro
;
Suzuki, Takayoshi
.
소스
In
Bioorganic & Medicinal Chemistry
15 January 2024 98
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7 . Academic Journal
Recent progress on small molecules targeting epigenetic complexes
저자
by
Itoh, Yukihiro
;
Takada, Yuri
;
Yamashita, Yasunobu
;
Suzuki, Takayoshi
.
소스
In
Current Opinion in Chemical Biology
April 2022 67
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6 . Academic Journal
Identification of a novel histone H2A mono-ubiquitination-inhibiting cell-active small molecule
저자
by
Ni, Siyao
;
Takada, Yuri
;
Ando, Takaaki
;
Yu, Shengwang
;
Yamashita, Yasunobu
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 June 2024 105
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7 . Academic Journal
Discovery of Selective Histone Deacetylase 1 and 2 Inhibitors: Screening of a Focused Library Constructed by Click Chemistry, Kinetic Binding Analysis, and Biological Evaluation.
저자
by
Itoh, Yukihiro
;
Zhan, Peng
;
Tojo, Toshifumi
;
Jaikhan, Pattaporn
;
Ota, Yosuke
, et al.
소스
Journal of Medicinal Chemistry; 11/23/2023, Vol. 66 Issue 22, p15171-15188, 18p
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7 . Academic Journal
Cancer-Cell-Selective Targeting by Arylcyclopropylamine–Vorinostat Conjugates.
저자
by
Ota, Yosuke
;
Itoh, Yukihiro
;
Kurohara, Takashi
;
Singh, Ritesh
;
Elboray, Elghareeb E.
, et al.
소스
ACS Medicinal Chemistry Letters; 10/13/2022, Vol. 13 Issue 10, p1568-1573, 6p
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7 . Academic Journal
Selective degradation of histone deacetylase 8 mediated by a proteolysis targeting chimera (PROTAC).
저자
by
Chotitumnavee, Jiranan
;
Yamashita, Yasunobu
;
Takahashi, Yukari
;
Takada, Yuri
;
Iida, Tetsuya
, et al.
소스
Chemical Communications
. 4/14/2022, Vol. 58 Issue 29, p4635-4638. 4p.
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7 . Academic Journal
Identification of Novel Histone Deacetylase 6‐Selective Inhibitors Bearing 3,3,3‐Trifluorolactic Amide (TFLAM) Motif as a Zinc Binding Group.
저자
by
Kurohara, Takashi
;
Tanaka, Keita
;
Takahashi, Daisuke
;
Ueda, Satoshi
;
Yamashita, Yasunobu
, et al.
소스
ChemBioChem; 11/16/2021, Vol. 22 Issue 22, p3158-3163, 6p
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7 . Periodical
Identification of Potent and Selective Inhibitors of Fat Mass Obesity-Associated Protein Using a Fragment-Merging Approach
저자
by
Prakash, Muthuraj
;
Itoh, Yukihiro
;
Fujiwara, Yoshie
;
Takahashi, Yukari
;
Takada, Yuri
, et al.
소스
Journal of Medicinal Chemistry; November 2021, Vol. 64 Issue: 21 p15810-15824, 15p
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7 . Academic Journal
Site-selective modification strategies in antibody–drug conjugates.
저자
by
Walsh, Stephen J.
;
Bargh, Jonathan D.
;
Dannheim, Friederike M.
;
Hanby, Abigail R.
;
Seki, Hikaru
, et al.
소스
Chemical Society Reviews
. 1/21/2021, Vol. 50 Issue 2, p1305-1353. 49p.
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