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1 . Academic Journal
Pharmacologic Evaluation of Orally Bioavailable Inhibitors of the 20S Proteasome.
저자
by
Kirk, Christopher J.
;
Aujay, Monette A.
;
Ho, Mark
;
Jiang, Jing
;
Laidig, Guy J.
, et al.
소스
In
Blood
16 November 2006 108(11):3581-3581
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7 . Academic Journal
The Novel, Irreversible Proteasome Inhibitor PR-171 Demonstrates Potent Anti-Tumor Activity in Pre-Clinical Models of Multiple Myeloma, and Overcomes Bortezomib Resistance.
저자
by
Kuhn, Deborah J.
;
Chen, Qing
;
Voorhees, Peter M.
;
Strader, John S.
;
Shenk, Kevin D.
, et al.
소스
In
Blood
16 November 2006 108(11):3461-3461
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7 . Academic Journal
Identification of Peptide Epoxy-Ketone Proteasome Inhibitors with Differential Active Site Selectivity.
저자
by
Demo, Susan D.
;
Aujay, Monette A.
;
Goldstein, Eileen
;
Laidig, Guy J.
;
Parlati, Francesco
, et al.
소스
In
Blood
16 November 2006 108(11):4398-4398
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7 . Academic Journal
Immunoproteasome-Selective Keto-Epoxide Inhibitors: Potential Therapeutic Agents for the Treatment of Hematological Disorders.
저자
by
Parlati, Francesco
;
Aujay, Monette A.
;
Demo, Susan D.
;
Goldstein, Eileen D.
;
Jiang, Jing
, et al.
소스
In
Blood
16 November 2006 108(11):4392-4392
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7 . Academic Journal
Biochemical and Cellular Characterization of the Novel Proteasome Inhibitor PR-171.
저자
by
Demo, Susan D.
;
Buchholz, Tonia J.
;
Laidig, Guy J.
;
Parlati, Francesco
;
Shenk, Kevin D.
, et al.
소스
In
Blood
16 November 2005 106(11):1588-1588
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7 . Academic Journal
Potent Activity of a Novel, Irreversible Inhibitor of the Ubiquitin-Proteasome Pathway Against Pre-Clinical Models of Multiple Myeloma.
저자
by
Kuhn, Deborah J.
;
Voorhees, Peter M.
;
Strader, John S.
;
Shenk, Kevin D.
;
Sun, Congcong M.
, et al.
소스
In
Blood
16 November 2005 106(11):1576-1576
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7 . Academic Journal
Pharmacokinetics, Pharmacodynamics and Anti-Tumor Efficacy of PR-171, a Novel Inhibitor of the 20S Proteasome.
저자
by
Kirk, Christopher J.
;
Bennett, Mark K.
;
Buchholz, Tonia J.
;
Demo, Susan D.
;
Ho, Mark N.
, et al.
소스
In
Blood
16 November 2005 106(11):609-609
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7 . Periodical
Potent activity of carfilzomib, a novel, irreversible inhibitor of the ubiquitin-proteasome pathway, against preclinical models of multiple myeloma
저자
by
Kuhn, Deborah J.
;
Chen, Qing
;
Voorhees, Peter M.
;
Strader, John S.
;
Shenk, Kevin D.
, et al.
소스
Blood; November 2007, Vol. 110 Issue: 9 p3281-3290, 10p
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7 . Academic Journal
Design and Synthesis of an Orally Bioavailable and Selective Peptide Epoxyketone Proteasome Inhibitor (PR-047)
저자
by
Zhou, Han-Jie
;
Aujay, Monette A.
;
Bennett, Mark K.
;
Dajee, Maya
;
Demo, Susan D.
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; MAY 14 2009, 52 9, p3028-p3038, 11p.
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7 . Academic Journal
Antitumor activity of PR-171, a novel irreversible inhibitor of the proteasome
저자
by
Demo, Susan D.
;
Kirk, Christopher J.
;
Aujay, Monette A.
;
Buchholz, Tonia J.
;
Dajee, Maya
, et al.
소스
CANCER RESEARCH
; JUL 1 2007, 67 13, p6383-p6391, 9p.
Full Text (AACR)
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