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1 . Academic Journal
A multidisciplinary study of 3-(β-d-glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: Computation, synthesis, crystallography and kinetics reveal new potent inhibitors
저자
by
Kun, Sándor
;
Begum, Jaida
;
Kyriakis, Efthimios
;
Stamati, Evgenia C.V.
;
Barkas, Thomas A.
, et al.
소스
In
European Journal of Medicinal Chemistry
10 March 2018 147:266-278
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7 . Academic Journal
Synthetic, enzyme kinetic, and protein crystallographic studies of C-β-d-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase
저자
by
Kantsadi, Anastassia L.
;
Bokor, Éva
;
Kun, Sándor
;
Stravodimos, George A.
;
Chatzileontiadou, Demetra S.M.
, et al.
소스
In
European Journal of Medicinal Chemistry
10 November 2016 123:737-745
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7 . Academic Journal
Biochemical and biological assessment of the inhibitory potency of extracts from vinification byproducts of Vitis vinifera extracts against glycogen phosphorylase
저자
by
Kantsadi, Anastassia L.
;
Apostolou, Anna
;
Theofanous, Stavroula
;
Stravodimos, George A.
;
Kyriakis, Efthimios
, et al.
소스
In
Food and Chemical Toxicology
May 2014 67:35-43
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7 . Academic Journal
Glucopyranosylidene-spiro-imidazolinones, a New Ring System: Synthesis and Evaluation as Glycogen Phosphorylase Inhibitors by Enzyme Kinetics and X‑ray Crystallography.
저자
by
Szabó, Katalin E.
;
Kyriakis, Efthimios
;
Psarra, Anna-Maria G.
;
Karra, Aikaterini G.
;
Sipos, Ádám
, et al.
소스
Journal of Medicinal Chemistry; 7/11/2019, Vol. 62 Issue 13, p6116-6136, 21p
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7 . Academic Journal
Probing the β-pocket of the active site of human liver glycogen phosphorylase with 3-(C-β-d-glucopyranosyl)-5-(4-substituted-phenyl)-1, 2, 4-triazole inhibitors.
저자
by
Kyriakis, Efthimios
;
Solovou, Theodora G.A.
;
Kun, Sándor
;
Czifrák, Katalin
;
Szőcs, Béla
, et al.
소스
Bioorganic Chemistry
. Apr2018, Vol. 77, p485-493. 9p.
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7 . Academic Journal
Nanomolar Inhibitors of Glycogen Phosphorylase Based on β-D-Glucosaminyl Heterocycles: A Combined Synthetic, Enzyme Kinetic, and Protein Crystallography Study.
저자
by
Bokor, Éva
;
Kyriakis, Efthimios
;
Solovou, Theodora G. A.
;
Koppány, Csenge
;
Kantsadi, Anastassia L.
, et al.
소스
Journal of Medicinal Chemistry
. 11/22/2017, Vol. 60 Issue 22, p9251-9262. 12p.
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7 . Academic Journal
van der Waals interactions govern C-β-d-glucopyranosyl triazoles’ nM inhibitory potency in human liver glycogen phosphorylase.
저자
by
Kantsadi, Anastassia L.
;
Stravodimos, George A.
;
Kyriakis, Efthimios
;
Chatzileontiadou, Demetra S.M.
;
Solovou, Theodora G.A.
, et al.
소스
Journal of Structural Biology
. Jul2017, Vol. 199 Issue 1, p57-67. 11p.
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7 . Academic Journal
Oxidation of human serum albumin exhibits inter-individual variability after an ultra-marathon mountain race.
저자
by
SPANIDIS, YPATIOS
;
PRIFTIS, ALEXANDROS
;
STAGOS, DIMITRIOS
;
STRAVODIMOS, GEORGE A.
;
LEONIDAS, DEMETRES D.
, et al.
소스
Experimental & Therapeutic Medicine
. May2017, Vol. 13 Issue 5, p2382-2390. 9p.
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7 . Periodical
Affinity Crystallography Reveals the Bioactive Compounds of Industrial Juicing Byproducts of Punica granatum for Glycogen Phosphorylase
저자
by
Stravodimos, George A.
;
Kantsadi, Anastassia L.
;
Apostolou, Anna
;
Kyriakis, Efthimios
;
Kafaski-Kanelli, Vassiliki-Nafsika
, et al.
소스
Current Drug Discovery Technologies; March 2018, Vol. 15 Issue: 1 p41-53, 13p
Full Text (Bentham Science)
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7 . Academic Journal
The ammonium sulfate inhibition of human angiogenin.
저자
by
Chatzileontiadou, Demetra S. M.
;
Tsirkone, Vicky G.
;
Dossi, Kyriaki
;
Kassouni, Aikaterini G.
;
Liggri, Panagiota G. V.
, et al.
소스
FEBS Letters
. Sep2016, Vol. 590 Issue 17, p3005-3018. 14p.
Web of Science
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