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1 .
Gold-Mediated Multiple Cysteine Arylation for the Construction of Highly Constrained Bicycle Peptides
저자
by
Gemma E. Mudd
;
Steven J. Stanway
;
David R. Witty
;
Alex Thomas
;
Silvia Baldo
, et al.
소스
Bioconjugate chemistry
. 33(8)
Scopus
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7 .
Influence of Lipophilicity on the Antibacterial Activity of Polymyxin Derivatives and on Their Ability to Act as Potentiators of Rifampicin
저자
by
Antoinette Wilson
;
Roy Lester
;
S. R. Moss
;
Mona Simonovic
;
Naomi Divall
, et al.
소스
ACS Infect Dis
Open Access (OpenAIRE)
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7 .
Direct modifications of the cyclic peptide Polymyxin B leading to analogues with enhanced in vitro antibacterial activity
저자
by
Pamela Brown
;
Steven Boakes
;
Steven J. Stanway
;
S. R. Moss
;
Antoinette Wilson
, et al.
소스
Bioorg Med Chem Lett
Open Access (OpenAIRE)
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7 . Academic Journal
Discovery of N-(3-Fluorophenyl)-1-[(4-([(3S)-3-methyl-1-piperazinyl]methyl)phenyl)acetyl]-4-piperidinamine (GSK962040), the First Small Molecule Motilin Receptor Agonist Clinical Candidate.
저자
by
Susan M. Westaway
;
Samantha L. Brown
;
Stephen C. M. Fell
;
Christopher N. Johnson
;
David T. MacPherson
, et al.
소스
Journal of Medicinal Chemistry
. Feb2009, Vol. 52 Issue 4, p1180-1189. 10p.
Full Text (ACS)
Web of Science
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7 .
Discovery of Potent Cyclophilin Inhibitors Based on the Structural Simplification of Sanglifehrin A
저자
by
Yu-Jen Lee
;
Andrew John Keats
;
Karine G. Poullennec
;
Uli Schmitz
;
Todd C. Appleby
, et al.
소스
Journal of Medicinal Chemistry
. 60:1000-1017
Web of Science
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7 .
Diastereoselective fluorination of silylated 1,2-oxazines to access fluorinated N,O-heterocycles
저자
by
Matthew N. Hopkinson
;
Steven J. Stanway
;
Véronique Gouverneur
;
Yu-hong Lam
.
소스
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6 .
1,5-Stereocontrol in tin(IV) halide mediated reactions between N- and S-substituted pent-2-enylstannanes and aldehydes or imines
저자
by
Eric J. Thomas
;
Steven J. Stanway
.
소스
Tetrahedron
. 68:5998-6009
Web of Science
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4 .
Recent progress in the use of fluoroorganic compounds in pericyclic reactions
저자
by
Véronique Gouverneur
;
Yu-hong Lam
;
Steven J. Stanway
.
소스
Tetrahedron
. 65:9905-9933
Open Access (OpenAIRE)
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5 .
Diels−Alder Exo Selectivity in Terminal-Substituted Dienes and Dienophiles: Experimental Discoveries and Computational Explanations
저자
by
Paul Ha-Yeon Cheong
;
José M. Blasco Mata
;
Véronique Gouverneur
;
Steven J. Stanway
;
Yu-hong Lam
, et al.
소스
Journal of the American Chemical Society
. 131:1947-1957
Open Access (OpenAIRE)
Web of Science
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7 .
The discovery of SB-435495
저자
by
V.Ann Lewis
;
Ian Stansfield
;
Kevin J. Milliner
;
Ivan Leo Pinto
;
Jackie C. Bloomer
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 12:2603-2606
Web of Science
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