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1 .
Agonist stimulation at human μ opioid receptors in a [(35)S]GTPγS incorporation assay: observation of 'bell-shaped' concentration-response relationships under conditions of strong receptor G protein coupling
저자
by
Didier Cussac
;
Stéphanie Tardif
;
Peter Heusler
.
소스
Journal of receptor and signal transduction research
. 36(2)
Scopus
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5 .
Pharmacological evaluation of a series of smoothened antagonists in signaling pathways and after topical application in a depilated mouse model
저자
by
Stéphanie Tardif
;
Amélie Tourette
;
David Troulier
;
Antoine Dumoulin
;
Marie‐Thérèse Calmettes
, et al.
소스
Pharmacology Research & Perspectives
Open Access (Wiley)
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7 .
The clozapine metabolite N-desmethylclozapine displays variable activity in diverse functional assays at human dopamine D2 and serotonin 5-HT1A receptors
저자
by
Stéphanie Tardif
;
Liesbeth A. Bruins Slot
;
Peter Heusler
;
Didier Cussac
;
Amélie Tourette
.
소스
European Journal of Pharmacology
. 669:51-58
Web of Science
Scopus
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7 .
Characterization of V0162, a new long-acting antagonist at human M3 muscarinic acetylcholine receptors
저자
by
Emmanuel Naline
;
Peter Heusler
;
Thierry Clerc
;
Didier Cussac
;
Stéphanie Tardif
, et al.
소스
Pharmacological research
. 100
Scopus
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7 .
Enhanced stability of wild-type and constitutively active α 2A -adrenoceptors by ligands with agonist, silent and inverse agonist properties
저자
by
Stéphanie Tardif
;
Petrus J. Pauwels
.
소스
Naunyn-Schmiedeberg's Archives of Pharmacology
. 366:134-141
Full Text (Springer)
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4 .
Differential signalling of both wild-type and Thr 343 Arg dopamine D 2short receptor by partial agonists in a G-protein-dependent manner 1 1Abbreviations: NPA, propylnorapomorphine; PTX, Bordetella pertussis toxin; 7-OH-DPAT, 7-(hydroxy-2-(di-n-propylamino)tetralin; and (+)-UH 232, cis-(+)-5-methoxy-1-methyl-2-(di-n-propylamino)tetralin
저자
by
Francis Colpaert
;
Stéphanie Tardif
;
Petrus J. Pauwels
.
소스
Biochemical Pharmacology
. 62:723-732
Web of Science
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5 .
Real-time analysis of dopamine: antagonist interactions at recombinant human D2longreceptor upon modulation of its activation state
저자
by
Stéphanie Tardif
;
Petrus J. Pauwels
;
Francis Colpaert
;
Thierry Wurch
.
소스
British Journal of Pharmacology
. 134:88-97
Full Text (Wiley)
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6 .
Modulation of 5-HT1A receptor signalling by point-mutation of cysteine351 in the rat Gαo protein
저자
by
Stéphanie Tardif
;
Petrus J. Pauwels
;
Thierry Wurch
;
Francis Colpaert
;
Delphine S. Dupuis
.
소스
Neuropharmacology
. 38:1035-1041
Web of Science
Scopus
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7 .
Stimulated [35S]GTPγS binding by 5-HT1A receptor agonists in recombinant cell lines Modulation of apparent efficacy by G-protein activation state
저자
by
Stéphanie Tardif
;
Francis Colpaert
;
P. J. Pauwels
;
Thierry Wurch
.
소스
Naunyn-Schmiedeberg's Archives of Pharmacology
. 356:551-561
Full Text (Springer)
Web of Science
Scopus
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6 .
[(3)H]-F13640, a novel, selective and high-efficacy serotonin 5-HT(1A) receptor agonist radioligand
저자
by
Stéphanie Tardif
;
Francis Colpaert
;
Christiane Palmier
;
Didier Cussac
;
Sophie Bernois
, et al.
소스
Naunyn-Schmiedeberg's archives of pharmacology
. 382(4)
Full Text (Springer)
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