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1 . Academic Journal
Methotrexate-based PROTACs as DHFR-specific chemical probes
저자
by
Rana, Sandeep
;
Dranchak, Patricia
;
Dahlin, Jayme L.
;
Lamy, Laurence
;
Li, Wenqing
, et al.
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In
Cell Chemical Biology
15 February 2024 31(2):221-233
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7 . Academic Journal
Discovering Targets of Non-enzymatic Acylation by Thioester Reactivity Profiling
저자
by
Kulkarni, Rhushikesh A.
;
Worth, Andrew J.
;
Zengeya, Thomas T.
;
Shrimp, Jonathan H.
;
Garlick, Julie M.
, et al.
소스
In
Cell Chemical Biology
16 February 2017 24(2):231-242
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7 . Academic Journal
Reference compounds for characterizing cellular injury in high-content cellular morphology assays
저자
by
Dahlin, Jayme L.
;
Hua, Bruce K.
;
Zucconi, Beth E.
;
Nelson, Jr, Shawn D.
;
Singh, Shantanu
, et al.
소스
Nature Communications
. 14(1)
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7 . Academic Journal
Suite of TMPRSS2 Assays for Screening Drug Repurposing Candidates as Potential Treatments of COVID-19.
저자
by
Shrimp, Jonathan H.
;
Janiszewski, John
;
Chen, Catherine Z.
;
Xu, Miao
;
Wilson, Kelli M.
, et al.
소스
ACS Infectious Diseases; 6/10/2022, Vol. 8 Issue 6, p1191-1203, 13p
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7 . Academic Journal
SULT1A1-dependent sulfonation of alkylators is a lineage-dependent vulnerability of liver cancers
저자
by
Shi, Lei
;
Shen, William
;
Davis, Mindy I.
;
Kong, Ke
;
Vu, Phuong
, et al.
소스
Nature Cancer
. 4(3):365-381
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7 . Academic Journal
Synergistic inhibition of SARS-CoV-2 cell entry by otamixaban and covalent protease inhibitors: pre-clinical assessment of pharmacological and molecular properties.
저자
by
Hempel, Tim
;
Elez, Katarina
;
Krüger, Nadine
;
Raich, Lluís
;
Shrimp, Jonathan H.
, et al.
소스
Chemical Science; 10/14/2021, Vol. 12 Issue 38, p12600-12609, 10p
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7 . Academic Journal
Discovery of TMPRSS2 Inhibitors from Virtual Screening as a Potential Treatment of COVID-19.
저자
by
Hu, Xin
;
Shrimp, Jonathan H.
;
Guo, Hui
;
Xu, Miao
;
Chen, Catherine Z.
, et al.
소스
ACS Pharmacology & Translational Science; 6/11/2021, Vol. 4 Issue 3, p1124-1135, 12p
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7 . Academic Journal
Remodelin Is a Cryptic Assay Interference Chemotype That Does Not Inhibit NAT10-Dependent Cytidine Acetylation.
저자
by
Shrimp, Jonathan H.
;
Jing, Yihang
;
Gamage, Supuni Thalalla
;
Nelson, Kathryn M.
;
Han, Joseph
, et al.
소스
ACS Medicinal Chemistry Letters; 6/10/2021, Vol. 12 Issue 6, p887-892, 6p
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7 . Academic Journal
An Enzymatic TMPRSS2 Assay for Assessment of Clinical Candidates and Discovery of Inhibitors as Potential Treatment of COVID-19.
저자
by
Shrimp, Jonathan H.
;
Kales, Stephen C.
;
Sanderson, Philip E.
;
Simeonov, Anton
;
Shen
, et al.
소스
ACS Pharmacology & Translational Science; 10/9/2020, Vol. 3 Issue 5, p997-1007, 11p
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7 . Periodical
Defining Metabolic and Nonmetabolic Regulation of Histone Acetylation by NSAID Chemotypes
저자
by
Shrimp, Jonathan H.
;
Garlick, Julie M.
;
Tezil, Tugsan
;
Sorum, Alexander W.
;
Worth, Andrew J.
, et al.
소스
Molecular Pharmaceutics; 20240101, Issue: Preprints
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