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1 . Academic Journal
Pharmacologic modulation of RNA splicing enhances anti-tumor immunity
저자
by
Lu, Sydney X.
;
De Neef, Emma
;
Thomas, James D.
;
Sabio, Erich
;
Rousseau, Benoit
, et al.
소스
In
Cell
22 July 2021 184(15):4032-4047
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7 . Academic Journal
Targeting PRMT1-mediated FLT3 methylation disrupts maintenance of MLL-rearranged acute lymphoblastic leukemia
저자
by
Zhu, Yinghui
;
He, Xin
;
Lin, Yi-Chun
;
Dong, Haojie
;
Zhang, Lei
, et al.
소스
In
Blood
10 October 2019 134(15):1257-1268
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7 . Academic Journal
PRMT1-mediated FLT3 arginine methylation promotes maintenance of FLT3-ITD+ acute myeloid leukemia
저자
by
He, Xin
;
Zhu, Yinghui
;
Lin, Yi-Chun
;
Li, Min
;
Du, Juan
, et al.
소스
In
Blood
8 August 2019 134(6):548-560
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7 . Academic Journal
Novel Allosteric Inhibitor-Derived AKT Proteolysis Targeting Chimeras (PROTACs) Enable Potent and Selective AKT Degradation in KRAS/BRAF Mutant Cells.
저자
by
Yu, Xufen
;
Xu, Jia
;
Cahuzac, Kaitlyn M.
;
Xie, Ling
;
Shen, Yudao
, et al.
소스
Journal of Medicinal Chemistry; 10/27/2022, Vol. 65 Issue 20, p14237-14260, 24p
Full Text (ACS)
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7 . Periodical
Dissecting and targeting noncanonical functions of EZH2 in multiple myeloma via an EZH2 degrader
저자
by
Yu, Xufen
;
Wang, Jun
;
Gong, Weida
;
Ma, Anqi
;
Shen, Yudao
, et al.
소스
Oncogene; March 2023, Vol. 42 Issue: 13 p994-1009, 16p
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7 . Academic Journal
Targeting Triple-Negative Breast Cancer by a Novel Proteolysis Targeting Chimera Degrader of Enhancer of Zeste Homolog 2.
저자
by
Dale, Brandon
;
Anderson, Chris
;
Park, Kwang-Su
;
Kaniskan, H. Ümit
;
Ma, Anqi
, et al.
소스
ACS Pharmacology & Translational Science; 7/8/2022, Vol. 5 Issue 7, p491-507, 17p
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7 . Academic Journal
Exploring Degradation of Mutant and Wild-Type Epidermal Growth Factor Receptors Induced by Proteolysis-Targeting Chimeras.
저자
by
Yu, Xufen
;
Cheng, Meng
;
Lu, Kaylene
;
Shen, Yudao
;
Zhong, Yue
, et al.
소스
Journal of Medicinal Chemistry; 6/23/2022, Vol. 65 Issue 12, p8416-8443, 28p
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7 . Periodical
PRMT inhibition induces a viral mimicry response in triple-negative breast cancer
저자
by
Wu, Qin
;
Nie, David Y.
;
Ba-alawi, Wail
;
Ji, YiShuai
;
Zhang, ZiWen
, et al.
소스
Nature Chemical Biology; August 2022, Vol. 18 Issue: 8 p821-830, 10p
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7 . Academic Journal
A selective WDR5 degrader inhibits acute myeloid leukemia in patient-derived mouse models.
저자
by
Yu, Xufen
;
Li, Dongxu
;
Kottur, Jithesh
;
Shen, Yudao
;
Kim, Huen Suk
, et al.
소스
Science Translational Medicine; 9/29/2021, Vol. 13 Issue 613, p1-16, 16p
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7 . Periodical
EZH2 noncanonically binds cMyc and p300 through a cryptic transactivation domain to mediate gene activation and promote oncogenesis
저자
by
Wang, Jun
;
Yu, Xufen
;
Gong, Weida
;
Liu, Xijuan
;
Park, Kwang-Su
, et al.
소스
Nature Cell Biology; March 2022, Vol. 24 Issue: 3 p384-399, 16p
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