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1 . Academic Journal
A 28-Day Toxicity Study of Tenofovir Alafenamide Hemifumarate by Subcutaneous Infusion in Rats and Dogs
저자
by
Doris Zane
;
Shane Roller
;
Josephine Shelton
;
Roshni Singh
;
Rachna Jain
, et al.
소스
Microbiology Spectrum, Vol 9, Iss 1 (2021)
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7 .
Tenofovir Alafenamide for HIV Prevention: Review of the Proceedings from the Gates Foundation Long-Acting TAF Product Development Meeting
저자
by
Zach R. Demkovich
;
Manjula Gunawardana
;
Ronald S. Veazey
;
Ariane van der Straten
;
Paul L. Feldman
, et al.
소스
AIDS Research and Human Retroviruses
Open Access (OpenAIRE)
Web of Science
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7 .
Abstract 2677: JZP815, a potent and selective pan-RAF inhibitor, demonstrates efficacy in RAF and RAS mutant tumor pre-clinical models
저자
by
Robert Hauptschein
;
Simon Woodcock
;
Andrew Belfield
;
Helen Mason
;
Dorottya Keppel
, et al.
소스
Cancer Research
. 82:2677-2677
Full Text (AACR)
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7 . Academic Journal
Discovery of the Dual Orexin Receptor Antagonist [(7R)-4-(5-Chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone (MK-4305) for the Treatment of Insomnia.
저자
by
Christopher D. Cox
;
Michael J. Breslin
;
David B. Whitman
;
John D. Schreier
;
Georgia B. McGaughey
, et al.
소스
Journal of Medicinal Chemistry
. Jul2010, Vol. 53 Issue 14, p5320-5332. 13p.
Full Text (ACS)
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7 .
Identification of potent, nonabsorbable agonists of the calcium-sensing receptor for GI-specific administration
저자
by
Lindsey T. Harston
;
David J. Cowan
;
Shane Roller
;
Caroline J. Diaz
;
Thomas J. Rimele
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 27:4673-4677
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7 .
ICA6150349, a Highly Selective Glucagon Agonist, in Combination with Exenatide Significantly Reduces Weight and Glucose in Obese and Diabetic Rats
저자
by
Mary K. Grizzle
;
Ved Srivastava
;
Rebecca J. Hodge
;
Mark A. Paulik
;
Andrew A. Young
, et al.
소스
Diabetes
. 67
Scopus
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7 .
Continuous Subcutaneous Delivery of a Glucagon Analog, ICA6150349, to Rats and Nonhuman Primates Demonstrates Safety and Tolerability in a 14-Day Toxicity Study
저자
by
Josephine Shelton
;
William Blackwell
;
Rebecca J. Hodge
;
Paul L. Feldman
;
Doris Zane
, et al.
소스
Diabetes
. 67
Scopus
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7 .
Exploration of phenylpropanoic acids as agonists of the free fatty acid receptor 4 (FFA4): Identification of an orally efficacious FFA4 agonist
저자
by
Erin Swiger
;
Thomas J. Rimele
;
Vincent Rash
;
David Moncol
;
Donald L. Hertzog
, et al.
소스
Bioorganicmedicinal chemistry letters
. 27(5)
Full Text (ScienceDirect)
Scopus
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7 .
Discovery of a Highly Potent, Nonabsorbable Apical Sodium-Dependent Bile Acid Transporter Inhibitor (GSK2330672) for Treatment of Type 2 Diabetes
저자
by
Eric E. Boros
;
Robert L. Dobbins
;
Maggie S. McIntyre
;
Ryan Klein
;
David J. Cowan
, et al.
소스
Journal of Medicinal Chemistry
. 56:5094-5114
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7 .
Orally bioavailable imidazoazepanes as calcitonin gene-related peptide (CGRP) receptor antagonists: Discovery of MK-2918
저자
by
Anthony W. Shaw
;
Theresa M. Williams
;
Joseph P. Vacca
;
Scott D. Mosser
;
Sean Yu
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 21:2683-2686
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