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1 . Academic Journal
A novel somatostatin receptor ligand for human ACTH – and GH –secreting pituitary adenomas.
저자
by
Regazzo, Daniela
;
Avallone, Serena
;
MacSweeney, Cliona P
;
Sergeev, Eugenia
;
Howe, David
, et al.
소스
European Journal of Endocrinology
. Jan2024, Vol. 190 Issue 1, pK8-K16. 9p.
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7 . Dissertation/ Thesis
Investigating the molecular pharmacology of the short chain fatty acid receptor FFA2
저자
by
Sergeev, Eugenia
.
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3 . Academic Journal
Targeting the Type 5 Metabotropic Glutamate Receptor: A Potential Therapeutic Strategy for Neurodegenerative Diseases?
저자
by
Budgett, Rebecca F.
;
Bakker, Geor
;
Sergeev, Eugenia
;
Bennett, Kirstie A.
;
Bradley, Sophie J.
.
소스
Frontiers in Pharmacology; 5/11/2022, Vol. 13, p1-20, 20p
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7 . Academic Journal
Structure‐Activity Relationship Explorations and Discovery of a Potent Antagonist for the Free Fatty Acid Receptor 2.
저자
by
Højgaard Hansen, Anders
;
Christensen, Henriette B.
;
Pandey, Sunil K.
;
Sergeev, Eugenia
;
Valentini, Alice
, et al.
소스
ChemMedChem; 11/5/2021, Vol. 16 Issue 21, p3326-3341, 16p
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7 . Periodical
Structure–Activity Relationship Studies of Tetrahydroquinolone Free Fatty Acid Receptor 3 Modulators
저자
by
Ulven, Elisabeth Rexen
;
Quon, Tezz
;
Sergeev, Eugenia
;
Barki, Natasja
;
Brvar, Matjaz
, et al.
소스
Journal of Medicinal Chemistry; April 2020, Vol. 63 Issue: 7 p3577-3595, 19p
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7 . Academic Journal
Discovery of a Potent Thiazolidine Free Fatty Acid Receptor 2 Agonist with Favorable Pharmacokinetic Properties.
저자
by
Hansen, Anders Højgaard
;
Sergeev, Eugenia
;
Bolognini, Daniele
;
Sprenger, Richard R.
;
Ekberg, Jeppe Hvidtfeldt
, et al.
소스
Journal of Medicinal Chemistry; 11/8/2018, Vol. 61 Issue 21, p9534-9550, 17p
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7 . Periodical
Chemogenetics defines receptor-mediated functions of short chain free fatty acids
저자
by
Bolognini, Daniele
;
Barki, Natasja
;
Butcher, Adrian
;
Hudson, Brian
;
Sergeev, Eugenia
, et al.
소스
Nature Chemical Biology; May 2019, Vol. 15 Issue: 5 p489-498, 10p
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7 . Academic Journal
Development and Characterization of a Fluorescent Tracer for the Free Fatty Acid Receptor 2 (FFA2/GPR43).
저자
by
Hansen, Anders Højgaard
;
Sergeev, Eugenia
;
Pandey, Sunil K.
;
Hudson, Brian D.
;
Christiansen, Elisabeth
, et al.
소스
Journal of Medicinal Chemistry
. Jul2017, Vol. 60 Issue 13, p5638-5645. 8p.
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7 . Academic Journal
A Novel Allosteric Activator of Free Fatty Acid 2 Receptor Displays Unique G
i
-functional Bias.
저자
by
Bolognini, Daniele
;
Moss, Catherine E.
;
Nilsson, Karolina
;
Petersson, Annika U.
;
Donnelly, Iona
, et al.
소스
Journal of Biological Chemistry
. 9/2/2016, Vol. 291 Issue 36, p18915-18931. 17p.
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7 . Academic Journal
Non-equivalence of Key Positively Charged Residues of the Free Fatty Acid 2 Receptor in the Recognition and Function of Agonist Versus Antagonist Ligands.
저자
by
Sergeev, Eugenia
;
Hansen, Anders Højgaard
;
Pandey, Sunil K.
;
MacKenzie, Amanda E.
;
Hudson, Brian D.
, et al.
소스
Journal of Biological Chemistry
. 1/1/2016, Vol. 291 Issue 1, p303-317. 15p.
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