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1 . Academic Journal
Biological and structural investigation of tetrahydro-β-carboline-based selective HDAC6 inhibitors with improved stability
저자
by
Scheuerer, Simon
;
Motlova, Lucia
;
Schäker-Hübner, Linda
;
Sellmer, Andreas
;
Feller, Felix
, et al.
소스
In
European Journal of Medicinal Chemistry
5 October 2024 276
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7 . Academic Journal
Identification of a highly efficient dual type I/II FMS-like tyrosine kinase inhibitor that disrupts the growth of leukemic cells
저자
by
Beyer, Mandy
;
Henninger, Sven J.
;
Haehnel, Patricia S.
;
Mustafa, Al-Hassan M.
;
Gurdal, Ece
, et al.
소스
In
Cell Chemical Biology
17 March 2022 29(3):398-411
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7 . Academic Journal
A novel Cereblon E3 ligase modulator with antitumor activity in gastrointestinal cancer
저자
by
Lier, Svenja
;
Sellmer, Andreas
;
Orben, Felix
;
Heinzlmeir, Stephanie
;
Krauß, Lukas
, et al.
소스
In
Bioorganic Chemistry
February 2022 119
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7 . Academic Journal
A series of novel aryl-methanone derivatives as inhibitors of FMS-like tyrosine kinase 3 (FLT3) in FLT3-ITD-positive acute myeloid leukemia
저자
by
Sellmer, Andreas
;
Pilsl, Bernadette
;
Beyer, Mandy
;
Pongratz, Herwig
;
Wirth, Lukas
, et al.
소스
In
European Journal of Medicinal Chemistry
1 May 2020 193
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7 . Academic Journal
Corrigendum to “A novel Cereblon E3 ligase modulator with antitumor activity in gastrointestinal cancer” [Bioorgan. Chem. 119 (2022) 105505]
저자
by
Lier, Svenja
;
Sellmer, Andreas
;
Orben, Felix
;
Heinzlmeir, Stephanie
;
Krauß, Lukas
, et al.
소스
In
Bioorganic Chemistry
May 2024 146
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7 . Academic Journal
Design and biological evaluation of tetrahydro-β-carboline derivatives as highly potent histone deacetylase 6 (HDAC6) inhibitors
저자
by
Leonhardt, Michel
;
Sellmer, Andreas
;
Krämer, Oliver H.
;
Dove, Stefan
;
Elz, Sigurd
, et al.
소스
In
European Journal of Medicinal Chemistry
25 May 2018 152:329-357
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7 . Academic Journal
Novel inhibitors of epidermal growth factor receptor: (4-(Arylamino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl)(1H-indol-2-yl)methanones and (1H-indol-2-yl)(4-(phenylamino)thieno[2,3-d]pyrimidin-6-yl)methanones
저자
by
Beckers, Thomas
;
Sellmer, Andreas
;
Eichhorn, Emerich
;
Pongratz, Herwig
;
Schächtele, Christoph
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 January 2012 20(1):125-136
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7 . Academic Journal
Inhibition of PDGFR tyrosine kinase activity by a series of novel N-(3-(4-(pyridin-3-yl)-1 H-imidazol-2-ylamino)phenyl)amides – A SAR study on the bioisosterism of pyrimidine and imidazole
저자
by
Mahboobi, Siavosh
;
Sellmer, Andreas
;
Eswayah, Asma
;
Elz, Sigurd
;
Uecker, Andrea
, et al.
소스
In
European Journal of Medicinal Chemistry
2008 43(7):1444-1453
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7 . Academic Journal
Antibacterial activity of a novel series of 3-bromo-4-(1 H-3-indolyl)-2,5-dihydro-1 H-2,5-pyrroledione derivatives – An extended structure–activity relationship study
저자
by
Mahboobi, Siavosh
;
Eichhorn, Emerich
;
Winkler, Matthias
;
Sellmer, Andreas
;
Möllmann, Ute
.
소스
In
European Journal of Medicinal Chemistry
2008 43(3):633-656
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7 . Academic Journal
Inhibition of FLT3 and PDGFR tyrosine kinase activity by bis(benzo[ b]furan-2-yl)methanones
저자
by
Mahboobi, Siavosh
;
Uecker, Andrea
;
Cénac, Christophe
;
Sellmer, Andreas
;
Eichhorn, Emerich
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2007 15(5):2187-2197
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