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1 . Academic Journal
Structure-Based Optimization of Selective and Brain Penetrant CK1δ Inhibitors for the Treatment of Circadian Disruptions.
저자
by
McCarver, Stefan
;
Hanna, Luke
;
Samant, Andrew
;
Thompson, Aaron A.
;
Seierstad, Mark
, et al.
소스
ACS Medicinal Chemistry Letters; 4/11/2024, Vol. 15 Issue 4, p486-492, 7p
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7 . Academic Journal
Convergent synthesis of thiodiazole dioxides from simple ketones and amines through an unusual nitrogen-migration mechanism.
저자
by
Punjajom, Kunlayanee
;
Sinclair, Paul P.
;
Saha, Ishika
;
Seierstad, Mark
;
Ameriks, Michael K.
, et al.
소스
Chemical Science; 1/7/2024, Vol. 15 Issue 1, p328-335, 8p
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7 . Academic Journal
Identification of highly selective SIK1/2 inhibitors that modulate innate immune activation and suppress intestinal inflammation.
저자
by
Babbe, Holger
;
Sundberg, Thomas B.
;
Tichenor, Mark
;
Seierstad, Mark
;
Bacani, Genesis
, et al.
소스
Proceedings of the National Academy of Sciences of the United States of America
. 1/2/2024, Vol. 121 Issue 1, p1-11. 49p.
Full Text (PNAS)
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7 . Academic Journal
Heteroarylureas with fused bicyclic diamine cores as inhibitors of fatty acid amide hydrolase
저자
by
Keith, John M.
;
Jones, William
;
Pierce, Joan M.
;
Seierstad, Mark
;
Palmer, James A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 October 2020 30(20)
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7 . Academic Journal
The SAR of brain penetration for a series of heteroaryl urea FAAH inhibitors
저자
by
Keith, John M.
;
Tichenor, Mark S.
;
Apodaca, Richard L.
;
Xiao, Wei
;
Jones, William M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 July 2016 26(13):3109-3114
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7 . Academic Journal
Novel Reagent Space: Identifying Unorderable but Readily Synthesizable Building Blocks.
저자
by
Seierstad, Mark
;
Tichenor, Mark S.
;
DesJarlais, Renee L.
;
Jim Na
;
Bacani, Genesis M.
, et al.
소스
ACS Medicinal Chemistry Letters; 11/11/2021, Vol. 12 Issue 11, p1853-1860, 8p
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7 . Academic Journal
1-Aryl-2-((6-aryl)pyrimidin-4-yl)amino)ethanols as competitive inhibitors of fatty acid amide hydrolase
저자
by
Keith, John M.
;
Hawryluk, Natalie
;
Apodaca, Richard L.
;
Chambers, Allison
;
Pierce, Joan M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 March 2014 24(5):1280-1284
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7 . Academic Journal
Heteroarylureas with spirocyclic diamine cores as inhibitors of fatty acid amide hydrolase
저자
by
Keith, John M.
;
Jones, William M.
;
Pierce, Joan M.
;
Seierstad, Mark
;
Palmer, James A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 February 2014 24(3):737-741
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7 . Academic Journal
Heteroaryl urea inhibitors of fatty acid amide hydrolase: Structure–mutagenicity relationships for arylamine metabolites
저자
by
Tichenor, Mark S.
;
Keith, John M.
;
Jones, William M.
;
Pierce, Joan M.
;
Merit, Jeff
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2012 22(24):7357-7362
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7 . Academic Journal
The discovery and synthesis of JNJ 31020028, a small molecule antagonist of the Neuropeptide Y Y2 receptor
저자
by
Swanson, Devin M.
;
Wong, Victoria D.
;
Jablonowski, Jill A.
;
Shah, Chandra
;
Rudolph, Dale A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 September 2011 21(18):5552-5556
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