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1 . Academic Journal
Finding the perfect spot for fluorine: Improving potency up to 40-fold during a rational fluorine scan of a Bruton’s Tyrosine Kinase (BTK) inhibitor scaffold
저자
by
Lou, Yan
;
Sweeney, Zachary K.
;
Kuglstatter, Andreas
;
Davis, Dana
;
Goldstein, David M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 January 2015 25(2):367-371
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7 . Academic Journal
Synthesis of Rovafovir Etalafenamide (Part I): Active Pharmaceutical Ingredient Process Development, Scale-Up, and Impurity Control Strategy.
저자
by
Standley, Eric A.
;
Bringley, Dustin A.
;
Calimsiz, Selcuk
;
Ng, Jeffrey D.
;
Sarma, Keshab
, et al.
소스
Organic Process Research & Development; 5/21/2021, Vol. 25 Issue 5, p1215-1236, 22p
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7 . Academic Journal
Synthesis of Rovafovir Etalafenamide (Part IV): Evolution of the Synthetic Process to the Fluorinated Nucleoside Fragment.
저자
by
Siler, David A.
;
Calimsiz, Selcuk
;
Doxsee, Ian J.
;
Kwong, Bernard
;
Ng, Jeffrey D.
, et al.
소스
Organic Process Research & Development; 5/21/2021, Vol. 25 Issue 5, p1263-1274, 12p
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7 . Academic Journal
Synthesis of Rovafovir Etalafenamide (Part II): Dynamic Control for Successful Scale-Up of an Oxygen-Releasing Elimination Reaction Mediated by Oxone.
저자
by
Bringley, Dustin A.
;
Roberts, Benjamin J.
;
Calimsiz, Selcuk
;
Brown, Brandon H.
;
Davy, Jason A.
, et al.
소스
Organic Process Research & Development; 5/21/2021, Vol. 25 Issue 5, p1237-1246, 10p
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7 . Academic Journal
Synthesis of Rovafovir Etalafenamide (Part III): Evolution of the Synthetic Process to the Phosphonamidate Fragment.
저자
by
Ambrosi, Andrea
;
Bringley, Dustin A.
;
Calimsiz, Selcuk
;
Garber, Jeffrey A. O.
;
Huynh, Huy
, et al.
소스
Organic Process Research & Development; 5/21/2021, Vol. 25 Issue 5, p1247-1262, 16p
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7 . Academic Journal
Isolation and identification of ester impurities in RG7128, an HCV polymerase inhibitor
저자
by
Chow, Justin
;
Liu, Yanzhou
;
Comstock, Kate
;
Brandl, Michael
;
Lin, Fangling
, et al.
소스
In
Journal of Pharmaceutical and Biomedical Analysis
2010 53(3):710-716
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7 . Academic Journal
Design, synthesis, and antiviral properties of 4′-substituted ribonucleosides as inhibitors of hepatitis C virus replication: The discovery of R1479
저자
by
Smith, David B.
;
Martin, Joseph A.
;
Klumpp, Klaus
;
Baker, Stewart J.
;
Blomgren, Peter A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2007 17(9):2570-2576
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7 . Academic Journal
Design and synthesis of orally active inhibitors of TNF synthesis as anti-rheumatoid arthritis drugs
저자
by
Chen, Jian Jeffrey
;
Dewdney, Nolan
;
Lin, Xiaohong
;
Martin, Robert L
;
Walker, Keith A.M
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2003 13(22):3951-3954
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7 . Academic Journal
Structure-Based Drug Designof RN486, a Potent andSelective Bruton’s Tyrosine Kinase (BTK) Inhibitor, for theTreatment of Rheumatoid Arthritis.
저자
by
Lou, Yan
;
Han, Xiaochun
;
Kuglstatter, Andreas
;
Kondru, Rama K.
;
Sweeney, Zachary K.
, et al.
소스
Journal of Medicinal Chemistry
. Jan2015, Vol. 58 Issue 1, p512-516. 5p.
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7 . Academic Journal
Design and Characterization of R1626, A Prodrug of the HCV Replication Inhibitor R1479 (4′-Azidocytidine) With Enhanced Oral Bioavailability
저자
by
Klumpp, Klaus
;
Smith, David
;
Brandl, Michael
;
Alfredson, Tom
;
Sarma, Keshab
, et al.
소스
In
Antiviral Research
2007 74(3):A35-A35
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