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1 . Periodical
Discovery and Preclinical Characterization of BIIB129, a Covalent, Selective, and Brain-Penetrant BTK Inhibitor for the Treatment of Multiple Sclerosis
저자
by
Himmelbauer, Martin K.
;
Bajrami, Bekim
;
Basile, Rebecca
;
Capacci, Andrew
;
Chen, TeYu
, et al.
소스
Journal of Medicinal Chemistry; May 2024, Vol. 67 Issue: 10 p8122-8140, 19p
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7 . Academic Journal
Corrigendum to “Optimization of a novel piperazinone series as potent selective peripheral covalent BTK inhibitors” [Bioorg. Med. Chem. Lett. 60 (2022) 128549]
저자
by
Ma, Bin
;
Metrick, Claire M.
;
Gu, Chungang
;
Hoemberger, Marc
;
Bajrami, Bekim
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 September 2022 72
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7 . Academic Journal
Optimization of a novel piperazinone series as potent selective peripheral covalent BTK inhibitors
저자
by
Ma, Bin
;
Metrick, Claire M.
;
Gu, Chungang
;
Hoemberger, Marc
;
Bajrami, Bekim
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 March 2022 60
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7 . Academic Journal
Colorimetric Detection of Glutamine Synthetase-Catalyzed Transferase Activity in Glucocorticoid-Treated Skeletal Muscle Cells
저자
by
Santoro, Joseph C.
;
Harris, Georgianna
;
Sitlani, Ayesha
.
소스
In
Analytical Biochemistry
1 February 2001 289(1):18-25
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5 . Academic Journal
Discovery of Potent, Selective, and Brain-Penetrant Apoptosis Signal-Regulating Kinase 1 (ASK1) Inhibitors that Modulate Brain Inflammation In Vivo.
저자
by
Jones, J. Howard
;
Zhili Xin
;
Himmelbauer, Martin
;
Dechantsreiter, Michael
;
Enyedy, Istvan
, et al.
소스
Journal of Medicinal Chemistry; 10/28/2021, Vol. 64 Issue 20, p15402-15419, 18p
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7 . Periodical
Discovery and Preclinical Characterization of BIIB091, a Reversible, Selective BTK Inhibitor for the Treatment of Multiple Sclerosis
저자
by
Hopkins, Brian T.
;
Bame, Eris
;
Bajrami, Bekim
;
Black, Cheryl
;
Bohnert, Tonika
, et al.
소스
Journal of Medicinal Chemistry; January 2022, Vol. 65 Issue: 2 p1206-1224, 19p
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7 . Academic Journal
Rational Design and Optimization of a Novel Class of Macrocyclic Apoptosis Signal-Regulating Kinase 1 Inhibitors.
저자
by
Himmelbauer, Martin K.
;
Xin, Zhili
;
Jones, J. Howard
;
Enyedy, Istvan
;
King, Kristopher
, et al.
소스
Journal of Medicinal Chemistry; 12/12/2019, Vol. 62 Issue 23, p10740-10756, 17p
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7 . Periodical
Human PLD structures enable drug design and characterization of isoenzyme selectivity
저자
by
Metrick, Claire M.
;
Peterson, Emily A.
;
Santoro, Joseph C.
;
Enyedy, Istvan J.
;
Murugan, Paramasivam
, et al.
소스
Nature Chemical Biology; April 2020, Vol. 16 Issue: 4 p391-399, 9p
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7 . Academic Journal
Novel ketal ligands for the glucocorticoid receptor: in vitro and in vivo activity
저자
by
Smith, Cameron J.
;
Ali, Amjad
;
Balkovec, James M.
;
Graham, Donald W.
;
Hammond, Milton L.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2005 15(11):2926-2931
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7 . Academic Journal
Discovery of CNS-Penetrant Apoptosis Signal-Regulating Kinase 1 (ASK1) Inhibitors
저자
by
Xin, Zhili
;
Himmelbauer, Martin K.
;
Jones, J. Howard
;
Enyedy, Istvan
;
Gilfillan, Rab
, et al.
소스
ACS MEDICINAL CHEMISTRY LETTERS
; APR 9 2020, 11 4, p485-p490, 6p.
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