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1 . Academic Journal
Pharmacological characterization of the ghrelin receptor antagonist, GSK1614343 in rat RC-4B/C cells natively expressing GHS type 1a receptors
저자
by
Perdonà, Elisabetta
;
Faggioni, Federico
;
Buson, Alberto
;
Sabbatini, Fabio Maria
;
Corti, Corrado
, et al.
소스
In
European Journal of Pharmacology
2011 650(1):178-183
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7 . Academic Journal
Synthesis and pharmacological characterisation of 2,4-Dicarboxy-pyrroles as selective non-Competitive mGluR1 antagonists
저자
by
Micheli, Fabrizio
;
Fabio, Romano Di
;
Cavanni, Paolo
;
Rimland, Joseph M
;
Capelli, Anna Maria
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2003 11(2):171-183
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7 . Academic Journal
Brain-penetrant cyanoindane and cyanotetralin inhibitors of G2019S-LRRK2 kinase activity.
저자
by
Garofalo, Albert W.
;
Schwarz, Jacob
;
Zobel, Kerry
;
Beato, Claudia
;
Bernardi, Silvia
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. Oct2023, Vol. 95, pN.PAG-N.PAG. 1p.
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7 . Academic Journal
Selective Inhibitors of G2019S-LRRK2 Kinase Activity.
저자
by
Garofalo, Albert W.
;
Bright, Jessica
;
De Lombaert, Stéphane
;
Toda, Alyssa M. A.
;
Zobel, Kerry
, et al.
소스
Journal of Medicinal Chemistry; 12/10/2020, Vol. 63 Issue 23, p14821-14839, 19p
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7 . Academic Journal
Design, synthesis and SAR of a novel series of benzimidazoles as potent NPY Y5 antagonists
저자
by
Pizzi, Domenica Antonia
;
Leslie, Colin Philip
;
Mazzali, Angelica
;
Seri, Catia
;
Biagetti, Matteo
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(23):7120-7123
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7 . Academic Journal
Novel substituted tetrahydrotriazaacenaphthylene derivatives as potent CRF 1 receptor antagonists
저자
by
Gentile, Gabriella
;
Di Fabio, Romano
;
Pavone, Francesca
;
Sabbatini, Fabio Maria
;
St-Denis, Yves
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2007 17(18):5218-5221
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7 . Academic Journal
From pyrroles to pyrrolo[1,2- a]pyrazinones: A new class of mGluR1 antagonists
저자
by
Micheli, Fabrizio
;
Cavanni, Paolo
;
Di Fabio, Romano
;
Marchioro, Carla
;
Donati, Daniele
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2006 16(5):1342-1345
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7 . Academic Journal
2,4-Dicarboxy-pyrroles as selective non-Competitive mGluR1 antagonists: further characterization of 3,5-Dimethyl pyrrole-2,4-dicarboxylic acid 2-propyl ester 4-(1,2,2-Trimethyl-propyl) ester and structure–Activity relationships
저자
by
Micheli, Fabrizio
;
Di Fabio, Romano
;
Bordi, Fabio
;
Cavallini, Palmina
;
Cavanni, Paolo
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2003 13(13):2113-2118
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7 . Academic Journal
Azabicyclo[3.1.0]hexane-1-carbohydrazides as Potent and Selective GHSR1a Ligands Presenting a Specific in vivo Behavior.
저자
by
Sabbatini, Fabio Maria
;
Melotto, Sergio
;
Bernasconi, Giovanni
;
Bromidge, Steve M.
;
D'Adamo, Lucilla
, et al.
소스
ChemMedChem; Nov2011, Vol. 6 Issue 11, p1981-1985, 5p
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7 . Academic Journal
Discovery Process and Characterization of Novel Carbohydrazide Derivatives as Potent and Selective GHSR1a Antagonists.
저자
by
Sabbatini, Fabio Maria
;
Di Fabio, Romano
;
Corsi, Mauro
;
Cavanni, Paolo
;
Bromidge, Steve M.
, et al.
소스
ChemMedChem; Sep2010, Vol. 5 Issue 9, p1450-1455, 6p
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