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1 .
Discovery of Two Novel Antiplatelet Clinical Candidates (BMS-986120 and BMS-986141) That Antagonize Protease-Activated Receptor 4
저자
by
E. Scott Priestley
;
Jacques Banville
;
Daniel Deon
;
Laurence Dubé
;
Marc Gagnon
, et al.
소스
Journal of Medicinal Chemistry
. 65:8843-8854
Web of Science
Scopus
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7 .
Discovery of Heteroaryl Urea Isosteres for Formyl Peptide Receptor 2 Agonists
저자
by
Nicholas R. Wurtz
;
James A. Johnson
;
Andrew Viet
;
Pravin S. Shirude
;
Vishweshwaraiah Baligar
, et al.
소스
ACS Med Chem Lett
Open Access (OpenAIRE)
Web of Science
Scopus
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7 .
Milvexian, an orally bioavailable, small‐molecule, reversible, direct inhibitor of factor XIa: In vitro studies and in vivo evaluation in experimental thrombosis in rabbits
저자
by
Jeffrey M. Bozarth
;
Pancras C. Wong
;
Earl J. Crain
;
William R. Ewing
;
Joseph M. Luettgen
, et al.
소스
Journal of Thrombosis and Haemostasis
. 20:399-408
Open Access (OpenAIRE)
Full Text (ScienceDirect O/A)
Web of Science
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7 .
Phthalazinone-Based Lactams and Cyclic Ureas as ROCK2 Selective Inhibitors
저자
by
Zilun Hu
;
Doree Sitkoff
;
Peter W. Glunz
;
Yan Zou
;
Cailan Wang
, et al.
소스
SSRN Electronic Journal
.
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7 .
Identification of a Hydroxypyrimidinone Compound (21) as a Potent APJ Receptor Agonist for the Potential Treatment of Heart Failure
저자
by
Wei Meng
;
Heather Finlay
;
Claudia Generaux
;
Chiuwa E. Luk
;
Tao Wang
, et al.
소스
Journal of Medicinal Chemistry
. 64:18102-18113
Web of Science
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7 .
Discussion of talks from the symposium: Factor X: From thrombokinase to oral anti-coagulants and beyond
저자
by
Ruth R. Wexler
;
Kenneth G. Mann
;
Leonard M. Milstone
;
Rodney M. Camire
;
Jeremy P. Wood
, et al.
소스
Journal of Thrombosis and Thrombolysis
Open Access (OpenAIRE)
Web of Science
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7 .
From basic science to life-saving therapy: the rationale, and drug discovery efforts that led to the direct factor Xa inhibitor eliquis
저자
by
Ruth R. Wexler
;
Robert M. Knabb
.
소스
Journal of Thrombosis and Thrombolysis
. 52:403-407
Web of Science
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4 .
Design and preparation of N-linked hydroxypyridine-based APJ agonists
저자
by
Jeremy M. Richter
;
J. Alex Bates
;
Peter Gargalovic
;
Joelle M. Onorato
;
Claudia Generaux
, et al.
소스
Bioorganicmedicinal chemistry letters
. 73
Scopus
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7 .
Discovery of a High Affinity, Orally Bioavailable Macrocyclic FXIa Inhibitor with Antithrombotic Activity in Preclinical Species
저자
by
Arunachalam Arumugam
;
Dietmar A. Seiffert
;
Arvind Mathur
;
Joanna J. Zheng
;
Ruth R. Wexler
, et al.
소스
Journal of Medicinal Chemistry
. 63:7226-7242
Web of Science
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7 .
Identification of 6-Hydroxypyrimidin-4(1H)-one-3-carboxamides as Potent and Orally Active APJ Receptor Agonists
저자
by
William A. Schumacher
;
Yan He
;
Peter S. Gargalovic
;
Tao Wang
;
Joelle M. Onorato
, et al.
소스
ACS Med Chem Lett
Open Access (OpenAIRE)
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