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1 . Academic Journal
Ligandability Assessment of IL-1β by Integrated Hit Identification Approaches.
저자
by
Vulpetti, Anna
;
Rondeau, Jean-Michel
;
Bellance, Marie-Hélène
;
Blank, Jutta
;
Boesch, Ralf
, et al.
소스
Journal of Medicinal Chemistry; 5/23/2024, Vol. 67 Issue 10, p8141-8160, 20p
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7 . Academic Journal
SEC-TID: A Label-Free Method for Small-Molecule Target Identification
저자
by
Salcius, Michael
;
Bauer, Andras J.
;
Hao, Qin
;
Li, Shu
;
Tutter, Antonin
, et al.
소스
In
SLAS Discovery
July 2014 19(6):917-927
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7 . Academic Journal
PIKfyve, a Class III PI Kinase, Is the Target of the Small Molecular IL-12/IL-23 Inhibitor Apilimod and a Player in Toll-like Receptor Signaling
저자
by
Cai, Xinming
;
Xu, Yongyao
;
Cheung, Atwood K.
;
Tomlinson, Ronald C.
;
Alcázar-Román, Abel
, et al.
소스
In
Chemistry & Biology
25 July 2013 20(7):912-921
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7 . Academic Journal
"Redirecting an anti-IL-1β antibody to bind a new, unrelated and computationally predicted epitope on hIL-17A".
저자
by
Fischman, Sharon
;
Levin, Itay
;
Rondeau, Jean-Michel
;
Štrajbl, Marek
;
Lehmann, Sylvie
, et al.
소스
Communications Biology
. 9/29/2023, Vol. 6 Issue 1, p1-13. 13p.
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7 . Academic Journal
Discovery of a selective and biologically active low-molecular weight antagonist of human interleukin-1β.
저자
by
Hommel, Ulrich
;
Hurth, Konstanze
;
Rondeau, Jean-Michel
;
Vulpetti, Anna
;
Ostermeier, Daniela
, et al.
소스
Nature Communications; 9/7/2023, Vol. 14 Issue 1, p1-13, 13p
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7 . Academic Journal
Discovery of amino-1,4-oxazines as potent BACE-1 inhibitors
저자
by
Veenstra, Siem Jakob
;
Rueeger, Heinrich
;
Voegtle, Markus
;
Lueoend, Rainer
;
Holzer, Philipp
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 July 2018 28(12):2195-2200
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7 . Academic Journal
Discovery of Umibecestat (CNP520): A Potent, Selective, and Efficacious β-Secretase (BACE1) Inhibitor for the Prevention of Alzheimer's Disease.
저자
by
Machauer, Rainer
;
Lueoend, Rainer
;
Hurth, Konstanze
;
Veenstra, Siem J.
;
Rueeger, Heinrich
, et al.
소스
Journal of Medicinal Chemistry; 10/28/2021, Vol. 64 Issue 20, p15262-15279, 18p
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7 . Book
Chapter 22 - Protein Crystallography and Drug Discovery
저자
by
Rondeau, Jean-Michel
;
Schreuder, Herman
.
소스
In
The Practice of Medicinal Chemistry
Edition: Fourth Edition. 2015:511-537
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4 . Academic Journal
Discovery of cyclic sulfoxide hydroxyethylamines as potent and selective β-site APP-cleaving enzyme 1 (BACE1) inhibitors: Structure based design and in vivo reduction of amyloid β-peptides
저자
by
Rueeger, Heinrich
;
Lueoend, Rainer
;
Machauer, Rainer
;
Veenstra, Siem Jacob
;
Jacobson, Laura Helen
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 October 2013 23(19):5300-5306
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7 . Periodical
Synthesis of the Potent, Selective, and Efficacious β-Secretase (BACE1) Inhibitor NB-360
저자
by
Rueeger, Heinrich
;
Lueoend, Rainer
;
Machauer, Rainer
;
Veenstra, Siem J.
;
Holzer, Philipp
, et al.
소스
Journal of Medicinal Chemistry; April 2021, Vol. 64 Issue: 8 p4677-4696, 20p
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