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1 . Academic Journal
Anticonvulsant profile of the neuroactive steroid, SGE-516, in animal models
저자
by
Hammond, Rebecca S.
;
Althaus, Alison L.
;
Ackley, Michael A.
;
Maciag, Carla
;
Martinez Botella, Gabriel
, et al.
소스
In
Epilepsy Research
August 2017 134:16-25
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7 . Academic Journal
Pharmacological characterization of SAGE‐718, a novel positive allosteric modulator of N‐methyl‐d‐aspartate receptors.
저자
by
Beckley, Jacob T.
;
Aman, Teresa K.
;
Ackley, Michael A.
;
Kazdoba, Tatiana M.
;
Lewis, Michael C.
, et al.
소스
British Journal of Pharmacology
. Apr2024, Vol. 181 Issue 7, p1028-1050. 23p.
Full Text (Wiley)
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7 . Academic Journal
Identification of 3-sulfonylindazole derivatives as potent and selective 5-HT6 antagonists
저자
by
Liu, Kevin G.
;
Robichaud, Albert J.
;
Greenfield, Alexander A.
;
Lo, Jennifer R.
;
Grosanu, Cristina
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 January 2011 19(1):650-662
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7 . Academic Journal
Di-substituted pyridinyl aminohydantoins as potent and highly selective human β-secretase (BACE1) inhibitors
저자
by
Malamas, Michael S.
;
Barnes, Keith
;
Johnson, Matthew
;
Hui, Yu
;
Zhou, Ping
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2010 18(2):630-639
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7 . Academic Journal
Dual acting norepinephrine reuptake inhibitors and 5-HT 2A receptor antagonists: Identification, synthesis and activity of novel 4-aminoethyl-3-(phenylsulfonyl)-1 H-indoles
저자
by
Heffernan, Gavin D.
;
Coghlan, Richard D.
;
Manas, Eric S.
;
McDevitt, Robert E.
;
Li, Yanfang
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2009 17(22):7802-7815
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7 . Academic Journal
3,4-Dihydropyrimido(1,2- a)indol-10(2 H)-ones as potent non-peptidic inhibitors of caspase-3
저자
by
Havran, Lisa M.
;
Chong, Dan C.
;
Childers, Wayne E.
;
Dollings, Paul J.
;
Dietrich, Arlene
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2009 17(22):7755-7768
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7 . Academic Journal
Novel 1-aminoethyl-3-arylsulfonyl-1 H-pyrrolo[2,3- b]pyridines are potent 5-HT 6 agonists
저자
by
Bernotas, Ronald C.
;
Lenicek, Steven
;
Antane, Schuyler
;
Cole, Derek C.
;
Harrison, Boyd L.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2009 17(14):5153-5163
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7 . Academic Journal
Novel 1-(azacyclyl)-3-arylsulfonyl-1 H-pyrrolo[2,3- b]pyridines as 5-HT 6 agonists and antagonists
저자
by
Elokdah, Hassan
;
Li, David
;
McFarlane, Geraldine
;
Bernotas, Ronald C.
;
Robichaud, Albert J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2007 15(18):6208-6226
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7 . Academic Journal
Novel neuroactive steroids as positive allosteric modulators of NMDA receptors: mechanism, site of action, and rescue pharmacology on GRIN variants associated with neurological conditions.
저자
by
Tang, Weiting
;
Beckley, Jacob T.
;
Zhang, Jin
;
Song, Rui
;
Xu, Yuchen
, et al.
소스
Cellular & Molecular Life Sciences
. Feb2023, Vol. 80 Issue 2, p1-20. 20p.
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7 . Academic Journal
SAGE-718: A First-in-Class N‑Methyl‑d‑Aspartate Receptor Positive Allosteric Modulator for the Potential Treatment of Cognitive Impairment.
저자
by
Hill, Matthew D.
;
Blanco, Maria-Jesus
;
Salituro, Francesco G.
;
Bai, Zhu
;
Beckley, Jacob T.
, et al.
소스
Journal of Medicinal Chemistry; 7/14/2022, Vol. 65 Issue 13, p9063-9075, 13p
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