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1 . Academic Journal
Discovery and Structure–Activity Relationship of Cadazolid: A First-In-Class Quinoxolidinone Antibiotic for the Treatment of Clostridioides difficile Infection.
저자
by
Rueedi, Georg
;
Panchaud, Philippe
;
Friedli, Astrid
;
Specklin, Jean-Luc
;
Hubschwerlen, Christian
, et al.
소스
Journal of Medicinal Chemistry; 6/13/2024, Vol. 67 Issue 11, p9465-9484, 20p
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7 . Academic Journal
Identification of SARS-CoV-2 Mpro inhibitors through deep reinforcement learning for de novo drug design and computational chemistry approaches.
저자
by
Hazemann, Julien
;
Kimmerlin, Thierry
;
Lange, Roland
;
Sweeney, Aengus Mac
;
Bourquin, Geoffroy
, et al.
소스
RSC Medicinal Chemistry; Jun2024, Vol. 15 Issue 6, p2146-2159, 14p
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7 . Academic Journal
Fragment‐based screening targeting an open form of the SARS‐CoV‐2 main protease binding pocket.
저자
by
Huang, Chia-Ying
;
Metz, Alexander
;
Lange, Roland
;
Artico, Nadia
;
Potot, Céline
, et al.
소스
Acta Crystallographica: Section D, Structural Biology
. Feb2024, Vol. 80 Issue 2, p123-136. 14p.
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7 . Periodical
Identification of SARS-CoV-2 Mpro inhibitors through deep reinforcement learning for de novodrug design and computational chemistry approachesElectronic supplementary information (ESI) available: The authors have cited additional references within the ESI.40–46See DOI: https://doi.org/10.1039/d4md00106k
저자
by
Hazemann, Julien
;
Kimmerlin, Thierry
;
Lange, Roland
;
Sweeney, Aengus Mac
;
Bourquin, Geoffroy
, et al.
소스
MedChemComm; 2024, Vol. 15 Issue: 6 p2146-2159, 14p
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7 . Academic Journal
Reduced IFN-ß inhibitory activity of Lagos bat virus phosphoproteins in human compared to Eidolon helvum bat cells.
저자
by
Papies, Jan
;
Sieberg, Andrea
;
Ritz, Daniel
;
Niemeyer, Daniela
;
Drosten, Christian
, et al.
소스
PLoS ONE
. 3/8/2022, Vol. 17 Issue 3, p1-20. 20p.
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7 . Academic Journal
Synthesis and Structure‐Activity Relationship of Xenocoumacin 1 and Analogues as Inhibitors of Ribosomal Protein Synthesis.
저자
by
Zumbrunn, Cornelia
;
Krüsi, Daniela
;
Stamm, Christina
;
Caspers, Patrick
;
Ritz, Daniel
, et al.
소스
ChemMedChem; 3/3/2021, Vol. 16 Issue 5, p891-897, 7p
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7 . Academic Journal
Structure-guided design, synthesis and biological evaluation of novel DNA ligase inhibitors with in vitro and in vivo anti-staphylococcal activity
저자
by
Surivet, Jean-Philippe
;
Lange, Roland
;
Hubschwerlen, Christian
;
Keck, Wolfgang
;
Specklin, Jean-Luc
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 November 2012 22(21):6705-6711
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7 . Academic Journal
Optimization of LpxC Inhibitor Lead Compounds Focusing on Efficacy and Formulation for High Dose Intravenous Administration.
저자
by
Panchaud, Philippe
;
Surivet, Jean-Philippe
;
Diethelm, Stefan
;
Blumstein, Anne-Catherine
;
Gauvin, Jean-Christophe
, et al.
소스
Journal of Medicinal Chemistry; 1/9/2020, Vol. 63 Issue 1, p88-102, 15p
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7 .
Nachhaltige Beziehungsgestaltung in der stationären Erziehungshilfe: Zur Bedeutung professioneller Bezugspersonenarbeit aus Sicht von Careleaver beim Übergang in die Selbstständigkeit
저자
by
Rippl, Melanie
;
Ritz, Daniel
.
소스
Open Access (OpenAIRE)
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4 . Periodical
Discovery of Novel Inhibitors of LpxC Displaying Potent in Vitro Activity against Gram-Negative Bacteria
저자
by
Surivet, Jean-Philippe
;
Panchaud, Philippe
;
Specklin, Jean-Luc
;
Diethelm, Stefan
;
Blumstein, Anne-Catherine
, et al.
소스
Journal of Medicinal Chemistry; May 2020, Vol. 63 Issue: 1 p66-87, 22p
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