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1 . Academic Journal
Synthesis, molecular modelling and QSAR study of new N-phenylacetamide-2-oxoindole benzensulfonamide conjugates as carbonic anhydrase inhibitors with antiproliferative activity
저자
by
Mona F. Said
;
Riham F. George
;
Andrea Petreni
;
Claudiu T. Supuran
;
Nada M. Mohamed
.
소스
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 701-717 (2022)
Open Access (DOAJ)
Open Access (T&F)
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7 . Academic Journal
Staquorsin: A Novel Staphylococcus aureus Agr-Mediated Quorum Sensing Inhibitor Impairing Virulence in vivo Without Notable Resistance Development
저자
by
Norhan H. Mahdally
;
Riham F. George
;
Mona T. Kashef
;
Medhat Al-Ghobashy
;
Fathia E. Murad
, et al.
소스
Frontiers in Microbiology, Vol 12 (2021)
Open Access (DOAJ)
Web of Science
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7 . Academic Journal
Aurones and furoaurones: Biological activities and synthesis
저자
by
Ghaneya S. Hassan
;
Hanan H. Georgey
;
Riham F. George
;
Eman R. Mohamed
.
소스
Bulletin of Faculty of Pharmacy Cairo University, Vol 56, Iss 2, Pp 121-127 (2018)
Full Text (ScienceDirect)
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6 .
Insights into targeting SARS-CoV-2: design, synthesis, in silico studies and antiviral evaluation of new dimethylxanthine derivatives
저자
by
Abdalla R. Mohamed
;
Ahmed Mostafa
;
Mahmoud A. El Hassab
;
Gomaa M. Hedeab
;
Sara H. Mahmoud
, et al.
소스
RSC Medicinal Chemistry
. 14:899-920
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7 .
Design, synthesis, in silico docking, ADMET and anticancer evaluations of thiazolidine-2,4-diones bearing heterocyclic rings as dual VEGFR-2/EGFRT790M tyrosine kinase inhibitors
저자
by
Nada A. A. M. Aziz
;
Riham F. George
;
Khaled El-Adl
;
Walaa R. Mahmoud
.
소스
RSC Advances
. 12:12913-12931
Open Access (OpenAIRE)
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6 .
Exploration of thiazolidine-2,4-diones as tyrosine kinase inhibitors: Design, synthesis, ADMET, docking, and antiproliferative evaluations
저자
by
Nada A. A. M. Aziz
;
Riham F. George
;
Khaled El‐Adl
;
Walaa R. Mahmoud
.
소스
Archiv der PharmazieREFERENCES
.
Scopus
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6 .
Design and synthesis of some new 6-bromo-2-(pyridin-3-yl)-4-substituted quinazolines as multi tyrosine kinase inhibitors
저자
by
Ahmed K.B.A.W. Farouk
;
Heba Abdelrasheed Allam
;
Essam Rashwan
;
Riham F. George
;
Safinaz E-S. Abbas
.
소스
Bioorganic chemistry
. 128
Scopus
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7 .
New benzimidazole derivatives targeting LasR with antibiofilm efficacy against Pseudomonas aeruginosa: An integrated in vitro and molecular dynamics simulation- based investigation
저자
by
Rehab H. Abd El-Aleam
;
Ahmed M. Sayed
;
Mostafa N. Taha
;
Riham F. George
;
Hanan H. Georgey
, et al.
소스
Journal of Molecular Structure
. 1277:134856
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7 .
Fluoroquinolone-3-carboxamide Amino Acid Conjugates: Synthesis, Antibacterial Properties And Molecular Modeling Studies
저자
by
Rajeev Sakhuja
;
Walid Fayad
;
Eatedal H. Abdel-Aal
;
Adel S. Girgis
;
Hitesh H. Honkanadavar
, et al.
소스
Medicinal Chemistry
. 17:71-84
Full Text (Bentham Science)
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7 .
HER2 Kinase-Targeted Breast Cancer Therapy: Design, Synthesis, and In Vitro and In Vivo Evaluation of Novel Lapatinib Congeners as Selective and Potent HER2 Inhibitors with Favorable Metabolic Stability
저자
by
Hamed I. Ali
;
Tamer A Elwaie
;
Safinaz E. Abbas
;
Enayat I. Aly
;
Khalid A. El Sayed
, et al.
소스
Journal of Medicinal Chemistry
. 63:15906-15945
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