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1 . Academic Journal
Exploration of the P1 residue in 3CL protease inhibitors leading to the discovery of a 2-tetrahydrofuran P1 replacement
저자
by
Barton, Linda S.
;
Callahan, James F.
;
Cantizani, Juan
;
Concha, Nestor O.
;
Cotillo Torrejon, Ignacio
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 February 2024 100
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7 . Academic Journal
A highly selective, cell-permeable furin inhibitor BOS-318 rescues key features of cystic fibrosis airway disease
저자
by
Douglas, Lisa E.J.
;
Reihill, James A.
;
Ho, Melisa W.Y.
;
Axten, Jeffrey M.
;
Campobasso, Nino
, et al.
소스
In
Cell Chemical Biology
16 June 2022 29(6):947-957
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7 . Academic Journal
Mechanistic MALDI-TOF Cell-Based Assay for the Discovery of Potent and Specific Fatty Acid Synthase Inhibitors
저자
by
Weigt, David
;
Parrish, Cynthia A.
;
Krueger, Julie A.
;
Oleykowski, Catherine A.
;
Rendina, Alan R.
, et al.
소스
In
Cell Chemical Biology
19 September 2019 26(9):1322-1331
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7 . Academic Journal
Orally bioavailable pyridine and pyrimidine-based Factor XIa inhibitors: Discovery of the methyl N-phenyl carbamate P2 prime group
저자
by
Corte, James R.
;
Fang, Tianan
;
Pinto, Donald J.P.
;
Orwat, Michael J.
;
Rendina, Alan R.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 May 2016 24(10):2257-2272
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7 . Academic Journal
Neutral macrocyclic factor VIIa inhibitors
저자
by
Wurtz, Nicholas R.
;
Parkhurst, Brandon L.
;
DeLucca, Indawati
;
Glunz, Peter W.
;
Jiang, Wen
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 June 2017 27(12):2650-2654
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7 . Academic Journal
Novel phenylalanine derived diamides as Factor XIa inhibitors
저자
by
Smith, Leon M., II
;
Orwat, Michael J.
;
Hu, Zilun
;
Han, Wei
;
Wang, Cailan
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 January 2016 26(2):472-478
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7 . Academic Journal
Structure-based design of inhibitors of coagulation factor XIa with novel P1 moieties
저자
by
Pinto, Donald J.P.
;
Smallheer, Joanne M.
;
Corte, James R.
;
Austin, Erin J.D.
;
Wang, Cailan
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 April 2015 25(7):1635-1642
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7 . Academic Journal
Pyridine and pyridinone-based factor XIa inhibitors
저자
by
Corte, James R.
;
Fang, Tianan
;
Hangeland, Jon J.
;
Friends, Todd J.
;
Rendina, Alan R.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 February 2015 25(4):925-930
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7 . Academic Journal
Orally bioavailable factor Xa inhibitors containing alpha-substituted gem-dimethyl P4 moieties
저자
by
Orwat, Michael J.
;
Qiao, Jennifer X.
;
He, Kan
;
Rendina, Alan R.
;
Luettgen, Joseph M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 August 2014 24(15):3341-3345
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7 . Academic Journal
Nonbenzamidine acylsulfonamide tissue factor–factor VIIa inhibitors
저자
by
Glunz, Peter W.
;
Zhang, Xiaojun
;
Zou, Yan
;
Delucca, Indawati
;
Nirschl, Alexandra H.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 September 2013 23(18):5244-5248
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