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1 . Academic Journal
Benzothienoquinazolinones as new multi-target scaffolds: Dual inhibition of human Topoisomerase I and tubulin polymerization
저자
by
Ceramella, Jessica
;
Caruso, Anna
;
Occhiuzzi, Maria Antonietta
;
Iacopetta, Domenico
;
Barbarossa, Alexia
, et al.
소스
In
European Journal of Medicinal Chemistry
1 November 2019 181
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7 . Academic Journal
Structure-guided design of pyridoclax derivatives based on Noxa / Mcl-1 interaction mode
저자
by
Hedir, Siham
;
De Giorgi, Marcella
;
Fogha, Jade
;
De Pascale, Martina
;
Weiswald, Louis-Bastien
, et al.
소스
In
European Journal of Medicinal Chemistry
5 November 2018 159:357-380
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7 . Academic Journal
Tau protein aggregation in Alzheimer's disease: An attractive target for the development of novel therapeutic agents
저자
by
Jouanne, Marie
;
Rault, Sylvain
;
Voisin-Chiret, Anne-Sophie
.
소스
In
European Journal of Medicinal Chemistry
20 October 2017 139:153-167
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5 . Academic Journal
Sequential one pot double C[sbnd]H heteroarylation of thiophene using bromopyridines to synthesize unsymmetrical 2,5-bipyridylthiophenes
저자
by
Kieffer, Charline
;
Babin, Victor
;
Jouanne, Marie
;
Slimani, Ikram
;
Berhault, Yohann
, et al.
소스
In
Tetrahedron
14 September 2017 73(37):5509-5516
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7 . Academic Journal
Multifaceted properties of 1,4-dimethylcarbazoles: Focus on trimethoxybenzamide and trimethoxyphenylurea derivatives as novel human topoisomerase II inhibitors
저자
by
Iacopetta, Domenico
;
Rosano, Camillo
;
Puoci, Francesco
;
Parisi, Ortensia Ilaria
;
Saturnino, Carmela
, et al.
소스
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European Journal of Pharmaceutical Sciences
1 January 2017 96:263-272
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7 . Academic Journal
3-(Dipropylamino)-5-hydroxybenzofuro[2,3-f]quinazolin-1(2H)-one (DPA-HBFQ-1) plays an inhibitory role on breast cancer cell growth and progression
저자
by
Rizza, Pietro
;
Pellegrino, Michele
;
Caruso, Anna
;
Iacopetta, Domenico
;
Sinicropi, Maria Stefania
, et al.
소스
In
European Journal of Medicinal Chemistry
1 January 2016 107:275-287
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7 . Academic Journal
Antileishmanial pharmacomodulation in 8-nitroquinolin-2(1H)-one series
저자
by
Kieffer, Charline
;
Cohen, Anita
;
Verhaeghe, Pierre
;
Paloque, Lucie
;
Hutter, Sébastien
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 May 2015 23(10):2377-2386
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7 . Academic Journal
Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium
저자
by
Cohen, Anita
;
Suzanne, Peggy
;
Lancelot, Jean-Charles
;
Verhaeghe, Pierre
;
Lesnard, Aurélien
, et al.
소스
In
European Journal of Medicinal Chemistry
5 May 2015 95:16-28
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7 . Academic Journal
Boronic species as promising inhibitors of the Staphylococcus aureus NorA efflux pump: Study of 6-substituted pyridine-3-boronic acid derivatives
저자
by
Fontaine, Fanny
;
Héquet, Arnaud
;
Voisin-Chiret, Anne-Sophie
;
Bouillon, Alexandre
;
Lesnard, Aurélien
, et al.
소스
In
European Journal of Medicinal Chemistry
5 May 2015 95:185-198
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7 . Academic Journal
Looking for new antileishmanial derivatives in 8-nitroquinolin-2(1H)-one series
저자
by
Kieffer, Charline
;
Cohen, Anita
;
Verhaeghe, Pierre
;
Hutter, Sébastien
;
Castera-Ducros, Caroline
, et al.
소스
In
European Journal of Medicinal Chemistry
6 March 2015 92:282-294
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