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1 .
Discovery of VNRX-7145 (VNRX-5236 Etzadroxil): An Orally Bioavailable β-Lactamase Inhibitor for Enterobacterales Expressing Ambler Class A, C, and D Enzymes
저자
by
William J. Weiss
;
Christopher J. Burns
;
Randy W. Jackson
;
Greg Moeck
;
Eugen F. Mesaros
, et al.
소스
Journal of Medicinal Chemistry
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7 .
Discovery of Taniborbactam (VNRX-5133): A Broad-Spectrum Serine- and Metallo-β-lactamase Inhibitor for Carbapenem-Resistant Bacterial Infections
저자
by
Bin Liu
;
M. Benvenuti
;
Christopher J. Burns
;
G.-H. Chu
;
Mcgarry Daniel G
, et al.
소스
'Journal of Medicinal Chemistry ', vol: 63, pages: 2789-2801 (2020)
Journal of Medicinal Chemistry
Open Access (OpenAIRE)
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7 .
VNRX-5133 (Taniborbactam), a broad-spectrum inhibitor of serine- And metallo-β-lactamases, restores activity of cefepime in enterobacterales and Pseudomonas aeruginosa
저자
by
Kaitlyn John
;
Jodie Hamrick
;
David A. Six
;
Denis M. Daigle
;
Tsuyoshi Uehara
, et al.
소스
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7 .
The discovery and structure–activity relationships of pyrano[3,4-b]indole-based inhibitors of hepatitis C virus NS5B polymerase
저자
by
Randy W. Jackson
;
Matthew G. LaPorte
;
Torsten Herbertz
;
Tandy L. Draper
;
Janet A. Gaboury
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 21:3227-3231
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7 .
The Discovery of Pyrano[3,4-b]indole-Based Allosteric Inhibitors of HCV NS5B Polymerase with In Vivo Activity
저자
by
Daniel C. Pevear
;
Dorothy C. Young
;
Christopher A. Benetatos
;
Glen A. Coburn
;
Susan R. Rippin
, et al.
소스
ChemMedChem
. 3:1508-1515
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7 .
Identification of TNF-α inhibitors from a split-Pool library based on a tyrosine-Proline peptidomimetic scaffold
저자
by
John C. Tabone
;
Randy W. Jackson
;
J. Jeffry Howbert
.
소스
Bioorganic & Medicinal Chemistry Letters
. 13:205-208
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5 .
Benzobicyclooctanes as novel inhibitors of TNF-α signaling
저자
by
J. Jeffry Howbert
;
Ted A. Baughman
;
John Latham
;
Devinder Singh
;
Thomas C. Cox
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 12:1093-1097
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7 .
Synthesis of a C-1 epi taxinine intermediate using the type 2 intramolecular Diels-Alder approach
저자
by
Kenneth J. Shea
;
Randy W. Jackson
.
소스
Tetrahedron Letters
. 35:1317-1320
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4 .
A mild and selective method for the cleavage of tert-butyl esters
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by
Randy W. Jackson
.
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Tetrahedron Letters
. 42:5163-5165
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3 .
ChemInform Abstract: The Chemistry of C-Aromatic Taxane Derivatives: Atropisomer Control of Reaction Stereochemistry
저자
by
Richard G. Higby
;
Randy W. Jackson
;
Jeffrey W. Gilman
;
Kenneth J. Shea
.
소스
ChemInform
. 23
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