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1 .
BMS-813160: A Potent CCR2 and CCR5 Dual Antagonist Selected as a Clinical Candidate
저자
by
Anne Rose
;
Qihong Zhao
;
Kumaravel Selvakumar
;
Percy H. Carter
;
Prakash Anjanappa
, et al.
소스
ACS Med Chem Lett
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7 .
Practical Synthesis of (3aR, 9bR)-8-Fluoro-7-(perfluoropropan-2-yl)-9b-(phenylsulfonyl)-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]indole: An Advanced Intermediate to Access the RORγt Inverse Agonist BMT-362265
저자
by
Manivel Pitchai
;
Anuradha Gupta
;
Arundutt Silamkoti
;
Amol G. Dikundwar
;
Prakash Anjanappa
, et al.
소스
Organic Process Research & Development
. 25:1001-1014
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Scopus
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7 .
Synthesis and characterization of a series of N,N′ ‐substituted urea derivatives by using electrospray ionization tandem mass spectrometry: Differentiation of positional isomers
저자
by
Sumit Kumar
;
Arvind Mathur
;
Venkatesh T. Kanthappa
;
Raju Gajjela
;
Arun Kumar Gupta
, et al.
소스
Rapid Communications in Mass Spectrometry
. 35
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7 .
Development of a Scalable Synthesis for the Potent Kinase Inhibitor BMS-986236; 1-(5-(4-(3-Hydroxy-3-methylbutyl)-1H-1,2,3-triazol-1-yl)-4-(isopropylamino)pyridin-2-yl)-1H-pyrazolo[3,4-b]pyridine-5-carbonitrile
저자
by
Lokesh Babu Jarugu
;
Suresh Krishnamoorthy
;
Anuradha Gupta
;
Muniyappa Shankar
;
Prakasam Kuppusamy
, et al.
소스
Organic Process Research & Development
. 23:912-918
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7 .
Discovery of a Hepatitis C Virus NS5B Replicase Palm Site Allosteric Inhibitor (BMS-929075) Advanced to Phase 1 Clinical Studies
저자
by
Katherine A. Grant-Young
;
Andrew Nickel
;
Rajesh Onkardas Bora
;
Prakash Anjanappa
;
Bender John A
, et al.
소스
Journal of Medicinal Chemistry
. 60:4369-4385
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7 .
Structure–Property Basis for Solving Transporter-Mediated Efflux and Pan-Genotypic Inhibition in HCV NS5B Inhibitors
저자
by
Hua Fang
;
Kevin Kish
;
Mark R. Witmer
;
Matthew G. Soars
;
Kyle Parcella
, et al.
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7 .
Carbamic acid 2-trimethylsilylethyl ester as a new ammonia equivalent for palladium-catalyzed amination of aryl halides
저자
by
Dibakar Mullick
;
Kandasamy Ruckmani
;
Manickam Sivakumar
;
Prakash Anjanappa
;
Kumaravel Selvakumar
.
소스
Tetrahedron Letters
. 51:5984-5987
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7 .
ChemInform Abstract: Carbamic Acid 2-Trimethylsilylethyl Ester as a New Ammonia Equivalent for Palladium-Catalyzed Amination of Aryl Halides
저자
by
Dibakar Mullick
;
Kandasamy Ruckmani
;
Manickam Sivakumar
;
Kumaravel Selvakumar
;
Prakash Anjanappa
.
소스
ChemInform
. 42
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7 .
ChemInform Abstract: 2-(Trimethylsilyl)ethanesulfonyl Amide as a New Ammonia Equivalent for Palladium-Catalyzed Amination of Aryl Halides
저자
by
Manickam Sivakumar
;
Kumaravel Selvakumar
;
Prakash Anjanappa
;
Dibakar Mullick
.
소스
ChemInform
. 39
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