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1 . Academic Journal
GSK114: A selective inhibitor for elucidating the biological role of TNNI3K
저자
by
Lawhorn, Brian G.
;
Philp, Joanne
;
Graves, Alan P.
;
Shewchuk, Lisa
;
Holt, Dennis A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 July 2016 26(14):3355-3358
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7 . Academic Journal
In vivo activity of an azole series of CCR2 antagonists
저자
by
Smethurst, Chris A.
;
Bevan, Nicola
;
Brooks, Carl
;
Emmons, Amanda
;
Gough, Peter J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2012 22(23):7252-7255
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7 . Academic Journal
Identification of a sulfonamide series of CCR2 antagonists
저자
by
Peace, Simon
;
Philp, Joanne
;
Brooks, Carl
;
Piercy, Val
;
Moores, Kitty
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(13):3961-3964
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7 . Academic Journal
The discovery of GSK221149A: A potent and selective oxytocin antagonist
저자
by
Liddle, John
;
Allen, Michael J.
;
Borthwick, Alan D.
;
Brooks, David P.
;
Davies, David E.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(1):90-94
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7 . Academic Journal
4,6-Diaminopyrimidines as Highly Preferred Troponin I-Interacting Kinase (TNNI3K) Inhibitors.
저자
by
Philp, Joanne
;
Lawhorn, Brian G.
;
Graves, Alan P.
;
Shewchuk, Lisa
;
Rivera, Katrina L.
, et al.
소스
Journal of Medicinal Chemistry
. 4/12/2018, Vol. 61 Issue 7, p3076-3088. 13p.
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7 . Academic Journal
Corrigendum to “In vivo activity of an azole series of CCR2 antagonists” [Bioorg. Med. Chem. Lett. 22 (2012) 7252–7255]
저자
by
Smethurst, Chris A.
;
Bevan, Nicola
;
Brooks, Carl
;
Emmons, Amanda
;
Gough, Peter J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 January 2013 23(1):382-382
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7 . Academic Journal
Substituent Effects on Drug-Receptor H-bond Interactions: Correlations Useful for the Design of Kinase Inhibitors.
저자
by
Lawhorn, Brian G.
;
Philp, Joanne
;
Graves, Alan P.
;
Holt, Dennis A.
;
Gatto Jr., Gregory J.
, et al.
소스
Journal of Medicinal Chemistry
. Dec2016, Vol. 59 Issue 23, p10629-10641. 13p.
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7 . Academic Journal
Inhibition of the Cardiomyocyte-Specific Kinase TNNI3K Limits Oxidative Stress, Injury, and Adverse Remodeling in the Ischemic Heart.
저자
by
Vagnozzi, Ronald J.
;
Gatto Jr., Gregory J.
;
Kallander, Lara S.
;
Hoffman, Nicholas E.
;
Mallilankaraman, Karthik
, et al.
소스
Science Translational Medicine; 10/16/2013, Vol. 5 Issue 207, p1-12, 12p
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7 . Academic Journal
Identification of Purines and 7-Deazapurines as Potent and Selective Type I Inhibitors of Troponin I-Interacting Kinase (TNNI3K)
저자
by
Lawhorn, Brian G.
;
Philp, Joanne
;
Zhao, Yongdong
;
Louer, Christopher
;
Hammond, Marlys
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; SEP 24 2015, 58 18, p7431-p7448, 18p.
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7 . Patent
저자
by
Kallander, Lara S.
;
Lawhorn, Brian Griffin
;
Philp, Joanne
;
Zhao, Yongdong
.
소스
Open Access (USPTO)
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