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1 . Academic Journal
Designing Selective Drug-like Molecular Glues for the Glucocorticoid Receptor/14-3‑3 Protein–Protein Interaction.
저자
by
Pallesen, Jakob S.
;
Munier, Claire C.
;
Bosica, Francesco
;
Andrei, Sebastian A.
;
Edman, Karl
, et al.
소스
Journal of Medicinal Chemistry; 12/22/2022, Vol. 65 Issue 24, p16818-16828, 11p
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7 . Academic Journal
Correction to "Designing Selective Drug-like Molecular Glues for the Glucocorticoid Receptor/14-3‑3 Protein–Protein Interaction".
저자
by
Pallesen, Jakob S.
;
Munier, Claire C.
;
Bosica, Francesco
;
Andrei, Sebastian A.
;
Edman, Karl
, et al.
소스
Journal of Medicinal Chemistry; 2/9/2023, Vol. 66 Issue 3, p2205-2207, 3p
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7 . Academic Journal
Glucocorticoid receptor Thr524 phosphorylation by MINK1 induces interactions with 14-3-3 protein regulators.
저자
by
Munier, Claire C.
;
De Maria, Leonardo
;
Edman, Karl
;
Gunnarsson, Anders
;
Longo, Marianna
, et al.
소스
Journal of Biological Chemistry
. Jan-Jun2021, Vol. 296, p1-15. 15p.
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7 . Periodical
Discovery of AZD8154, a Dual PI3Kγδ Inhibitor for the Treatment of Asthma
저자
by
Perry, Matthew W. D.
;
Björhall, Karin
;
Bold, Peter
;
Brűlls, Mikael
;
Börjesson, Ulf
, et al.
소스
Journal of Medicinal Chemistry; June 2021, Vol. 64 Issue: 12 p8053-8075, 23p
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7 . Academic Journal
Design, Synthesis, and Biological Evaluation of MEK PROTACs.
저자
by
Vollmer, Stefan
;
Cunoosamy, Danen
;
Lv, Huafei
;
Feng, Huanxi
;
Li, Xia
, et al.
소스
Journal of Medicinal Chemistry; 1/9/2020, Vol. 63 Issue 1, p157-162, 6p
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7 . Periodical
PI3K inhibitors are finally coming of age
저자
by
Vanhaesebroeck, Bart
;
Perry, Matthew W. D.
;
Brown, Jennifer R.
;
André, Fabrice
;
Okkenhaug, Klaus
.
소스
Nature Reviews Drug Discovery; 20210101, Issue: Preprints p1-29, 29p
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7 . Periodical
Identification of Phosphate-Containing Compounds as New Inhibitors of 14-3-3/c-Abl Protein–Protein Interaction
저자
by
Iralde-Lorente, Leire
;
Tassone, Giusy
;
Clementi, Letizia
;
Franci, Lorenzo
;
Munier, Claire C
, et al.
소스
ACS Chemical Biology; April 2020, Vol. 15 Issue: 4 p1026-1035, 10p
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7 . Academic Journal
Evolution of PI3Kγ and δ Inhibitors for Inflammatory and Autoimmune Diseases.
저자
by
Perry, Matthew W. D.
;
Abdulai, Raolat
;
Mogemark, Mickael
;
Petersen, Jens
;
Thomas, Matthew J.
, et al.
소스
Journal of Medicinal Chemistry; 5/23/2019, Vol. 62 Issue 10, p4783-4814, 32p
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7 . Academic Journal
Discovery of Highly Isoform Selective Orally Bioavailable Phosphoinositide 3‑Kinase (PI3K)‑γ Inhibitors.
저자
by
Pemberton, Nils
;
Mogemark, Mickael
;
Arlbrandt, Susanne
;
Bold, Peter
;
Cox, Rhona J.
, et al.
소스
Journal of Medicinal Chemistry; 6/28/2018, Vol. 61 Issue 12, p5435-5441, 7p
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7 . Periodical
A class of highly selective inhibitors bind to an active state of PI3Kγ
저자
by
Gangadhara, Gangadhara
;
Dahl, Göran
;
Bohnacker, Thomas
;
Rae, Rebecca
;
Gunnarsson, Jenny
, et al.
소스
Nature Chemical Biology; April 2019, Vol. 15 Issue: 4 p348-357, 10p
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