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1 . Academic Journal
A small-molecule inhibitor of the BRCA2-RAD51 interaction modulates RAD51 assembly and potentiates DNA damage-induced cell death
저자
by
Scott, Duncan E.
;
Francis-Newton, Nicola J.
;
Marsh, May E.
;
Coyne, Anthony G.
;
Fischer, Gerhard
, et al.
소스
In
Cell Chemical Biology
17 June 2021 28(6):835-847
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7 . Academic Journal
Releasing the technical ‘shackles’ on GPCR drug discovery: opportunities enabled by detergent-free polymer lipid particle (PoLiPa) purification
저자
by
Hothersall, J. Daniel
;
Jones, Andrew Y.
;
Dafforn, Tim R.
;
Perrior, Trevor
;
Chapman, Kathryn L.
.
소스
In
Drug Discovery Today
November 2020 25(11):1944-1956
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7 . Dissertation/ Thesis
Targeting IKKε/TBK1 for the treatment of diffuse large B-cell lymphoma
저자
by
Carr, Matthew D.
;
Perrior, Trevor
;
Chapman, Katie
.
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5 . Academic Journal
Stereoselective electrophile-induced mono- and bis-cyclisation–fragmentation reactions of alkenyl oxime O-allyl and O-benzyl ethers. Synthesis of dihydropinidine
저자
by
Ali Dondas, H
;
Grigg, Ronald
;
Markandu, Jasothara
;
Perrior, Trevor
;
Suzuki, Tekka
, et al.
소스
In
Tetrahedron
2002 58(1):161-173
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7 . Academic Journal
Preclinical trial of a MAP4K4 inhibitor to reduce infarct size in the pig: does cardioprotection in human stem cell‑derived myocytes predict success in large mammals?
저자
by
te Lintel Hekkert, Maaike
;
Newton, Gary
;
Chapman, Kathryn
;
Aqil, Rehan
;
Downham, Robert
, et al.
소스
Basic Research in Cardiology
. Jan2021, Vol. 116 Issue 1, p1-12. 12p. 4 Graphs.
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7 . Academic Journal
IKKε and TBK1 in diffuse large B‐cell lymphoma: A possible mechanism of action of an IKKε/TBK1 inhibitor to repress NF‐κB and IL‐10 signalling.
저자
by
Carr, Matthew
;
Mamand, Sami
;
Chapman, Kathryn L.
;
Perrior, Trevor
;
Wagner, Simon D.
.
소스
Journal of Cellular & Molecular Medicine; Oct2020, Vol. 24 Issue 19, p11573-11582, 10p
Open Access (Wiley)
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7 . Academic Journal
Selective protection of human cardiomyocytes from anthracycline cardiotoxicity by small molecule inhibitors of MAP4K4.
저자
by
Golforoush, Pelin A.
;
Narasimhan, Priyanka
;
Chaves-Guerrero, Patricia P.
;
Lawrence, Elsa
;
Newton, Gary
, et al.
소스
Scientific Reports
. 7/21/2020, Vol. 10 Issue 1, p1-12. 12p.
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7 . Academic Journal
IKK epsilon and TBK1 in diffuse large B-cell lymphoma: A possible mechanism of action of an IKK epsilon/TBK1 inhibitor to repress NF-kappa B and IL-10 signalling
저자
by
Carr, Matthew
;
Mamand, Sami
;
Chapman, Kathryn L.
;
Perrior, Trevor
;
Wagner, Simon D.
.
소스
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE
; OCT 2020, 24 19, p11573-p11582, 10p.
Open Access (Wiley)
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7 . Academic Journal
Design and discovery of 3-aryl-5-substituted-isoquinolin-1-ones as potent tankyrase inhibitors.
저자
by
Elliott, Richard J. R.
;
Jarvis, Ashley
;
Rajasekaran, Mohan B.
;
Menon, Malini
;
Bowers, Leandra
, et al.
소스
MedChemComm; Sep2015, Vol. 6 Issue 9, p1687-1692, 6p
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7 . Periodical
Generation and Trapping of Acyl Nitrile Oxides from Substituted Aryl 1,3 Diketones in a Nitrating Mixture
저자
by
Barrett, David
;
Bentley, Philip
;
Perrior, Trevor
.
소스
Synthetic Communications; September 1996, Vol. 26 Issue: 18 p3401-3406, 6p
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