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1 . Academic Journal
Minor chemical modifications of the aminosteroid derivative RM-581 lead to major impact on its anticancer activity, metabolic stability and aqueous solubility
저자
by
Maltais, René
;
Perreault, Martin
;
Roy, Jenny
;
Poirier, Donald
.
소스
In
European Journal of Medicinal Chemistry
15 February 2020 188
Full Text (ScienceDirect)
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6 . Academic Journal
Synthesis and evaluation of substituted phenyl cycloalkylureas and bioisosteres as IL-6 expression inhibitors.
저자
by
Tremblay, Sébastien
;
Boutin, Joël
;
Perreault, Martin
;
Côté, Marie-France
;
Gobeil, Stéphane
, et al.
소스
Medicinal Chemistry Research; Aug2020, Vol. 29 Issue 8, p1424-1437, 14p
Web of Science
Scopus
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7 . Academic Journal
A- and D‑Ring Structural Modifications of an Androsterone Derivative Inhibiting 17β-Hydroxysteroid Dehydrogenase Type 3: Chemical Synthesis and Structure–Activity Relationships.
저자
by
Cortés-Benítez, Francisco
;
Roy, Jenny
;
Perreault, Martin
;
Maltais, René
;
Poirier, Donald
.
소스
Journal of Medicinal Chemistry; 8/8/2019, Vol. 62 Issue 15, p7070-7088, 19p
Full Text (ACS)
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7 . Academic Journal
Induction of endoplasmic reticulum stress by aminosteroid derivative RM-581 leads to tumor regression in PANC-1 xenograft model.
저자
by
Perreault, Martin
;
Maltais, René
;
Roy, Jenny
;
Picard, Sylvain
;
Popa, Ion
, et al.
소스
Investigational New Drugs; Jun2019, Vol. 37 Issue 3, p431-440, 10p
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7 . Academic Journal
Urinary Elimination of Bile Acid Glucuronides under Severe Cholestatic Situations: Contribution of Hepatic and Renal Glucuronidation Reactions.
저자
by
Perreault, Martin
;
Wunsch, Ewa
;
Białek, Andrzej
;
Trottier, Jocelyn
;
Verreault, Mélanie
, et al.
소스
Canadian Journal of Gastroenterology & Hepatology; 4/11/2018, p1-12, 12p
Open Access (Wiley)
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7 . Academic Journal
Implication of STARD5 and cholesterol homeostasis disturbance in the endoplasmic reticulum stress-related response induced by pro-apoptotic aminosteroid RM-133.
저자
by
Perreault, Martin
;
Maltais, René
;
Kenmogne, Lucie Carolle
;
Létourneau, Danny
;
LeHoux, Jean-Guy
, et al.
소스
Pharmacological Research
. Feb2018, Vol. 128, p52-60. 9p.
Full Text (ScienceDirect)
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7 . Academic Journal
Insight into the mode of action and selectivity of PBRM, a covalent steroidal inhibitor of 17β-hydroxysteroid dehydrogenase type 1.
저자
by
Trottier, Alexandre
;
Maltais, René
;
Ayan, Diana
;
Barbeau, Xavier
;
Roy, Jenny
, et al.
소스
Biochemical Pharmacology
. Nov2017, Vol. 144, p149-161. 13p.
Full Text (ScienceDirect)
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7 . Academic Journal
Design of a Mestranol 2- N-Piperazino-Substituted Derivative Showing Potent and Selective in vitro and in vivo Activities in MCF-7 Breast Cancer Models.
저자
by
Perreault, Martin
;
Maltais, René
;
Roy, Jenny
;
Dutour, Raphaël
;
Poirier, Donald
.
소스
ChemMedChem; 1/20/2017, Vol. 12 Issue 2, p177-182, 6p
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7 . Academic Journal
Explorative study on the anticancer activity, selectivity and metabolic stability of related analogs of aminosteroid RM-133.
저자
by
Perreault, Martin
;
Maltais, René
;
Dutour, Raphaël
;
Poirier, Donald
.
소스
Steroids
. Nov2016, Vol. 115, p105-113. 9p.
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6 . Periodical
Parallel Solid-Phase Synthesis using a New Diethylsilylacetylenic Linker and Leading to Mestranol Derivatives with Potent Antiproliferative Activities on Multiple Cancer Cell Lines
저자
by
Dutour, Raphaël
;
Maltais, René
;
Perreault, Martin
;
Roy, Jenny
;
Poirier, Donald
.
소스
Anti-Cancer Agents in Medicinal Chemistry; August 2018, Vol. 18 Issue: 10 p1469-1481, 13p
Full Text (Bentham Science)
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