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1 . Academic Journal
Rapid Lentiviral Vector Producer Cell Line Generation Using a Single DNA Construct
저자
by
Yu Hua Chen
;
Celeste Pallant
;
Christopher J. Sampson
;
Alessia Boiti
;
Sabine Johnson
, et al.
소스
Molecular Therapy: Methods & Clinical Development, Vol 19, Iss , Pp 47-57 (2020)
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7 .
Rapid Lentiviral Vector Producer Cell Line Generation Using a Single DNA Construct
저자
by
P. Hardwicke
;
Christopher J. Sampson
;
Martijn H. Brugman
;
Cindy Jung
;
Yu Hua Chen
, et al.
소스
Molecular Therapy: Methods & Clinical Development, Vol 19, Iss, Pp 47-57 (2020)
Molecular Therapy. Methods & Clinical Development
Full Text (ScienceDirect O/A)
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7 . Academic Journal
The Discovery ofin Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm)Inhibitors by Hybridizing Fragment and HTS Hits.
저자
by
Sophie M. Bertrand
;
Nicolas Ancellin
;
Benjamin Beaufils
;
Ryan P. Bingham
;
Jennifer A. Borthwick
, et al.
소스
Journal of Medicinal Chemistry
. Sep2015, Vol. 58 Issue 18, p7140-7163. 24p.
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7 .
Catalytic in vivo protein knockdown by small-molecule PROTACs
저자
by
Natasha Routly
;
Giovanna Bergamini
;
Jeffrey L. Gustafson
;
Ko Eunhwa
;
Kristoffer Famm
, et al.
소스
Nature Chemical Biology
. 11:611-617
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7 .
Structurally diverse mitochondrial branched chain aminotransferase (BCATm) leads with varying binding modes identified by fragment screening
저자
by
Colin J. Suckling
;
Claus Spitzfaden
;
Andrew N. Hobbs
;
Craig Jamieson
;
Peter Francis
, et al.
소스
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7 .
Discovery and Optimization of Potent, Selective, and in Vivo Efficacious 2-Aryl Benzimidazole BCATm Inhibitors
저자
by
Svetlana L. Belyanskaya
;
Chun-wa Chung
;
Eric Humphries
;
Christopher S. Kollmann
;
Nicolas Ancellin
, et al.
소스
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7 .
Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitor
저자
by
Philip Alan Skone
;
Donald O. Somers
;
Marion C. Dickson
;
Nick Smithers
;
Ann Louise Walker
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 21:6188-6194
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7 .
Kinetic assay for characterization of spleen tyrosine kinase activity and inhibition with recombinant kinase and crude cell lysates
저자
by
Angela M. Deakin
;
Erik Schaefer
;
Paolo Luraghi
;
Min Li
;
Clare I. Hobbs
, et al.
소스
Analytical Biochemistry
. 384:56-67
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7 .
Discovery, SAR, and X-ray Binding Mode Study of BCATm Inhibitors from a Novel DNA-Encoded Library
저자
by
Laura J Pothier Kaushansky
;
Jennifer L. DeLorey
;
Hongfeng Deng
;
Christopher P. Davie
;
Jingye Zhou
, et al.
소스
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7 .
The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits
저자
by
Ian Churcher
;
Sarah E. Smith
;
Ryan P. Bingham
;
Clare I. Hobbs
;
Donald O. Somers
, et al.
소스
Journal of medicinal chemistry
. 58(18)
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