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1 . Academic Journal
Structural and mechanistic basis of differentiated inhibitors of the acute pancreatitis target kynurenine-3-monooxygenase
저자
by
Jonathan P. Hutchinson
;
Paul Rowland
;
Mark R. D. Taylor
;
Erica M. Christodoulou
;
Carl Haslam
, et al.
소스
Nature Communications, Vol 8, Iss 1, Pp 1-12 (2017)
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7 .
Investigation of Janus Kinase (JAK) Inhibitors for Lung Delivery and the Importance of Aldehyde Oxidase Metabolism
저자
by
Christopher R. Wellaway
;
Ian R. Baldwin
;
Paul Bamborough
;
Daniel Barker
;
Michelle A. Bartholomew
, et al.
소스
Journal of Medicinal Chemistry
. 65:633-664
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7 .
Optimization of Orally Bioavailable PI3Kδ Inhibitors and Identification of Vps34 as a Key Selectivity Target
저자
by
Giovanna Bergamini
;
Stefano Livia
;
Kenneth David Down
;
Marcus Bantscheff
;
Nick Barton
, et al.
소스
Journal of Medicinal Chemistry
. 63:638-655
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7 .
Mechanism for antigenic peptide selection by endoplasmic reticulum aminopeptidase 1
저자
by
Paraskevi Kokkala
;
Aggelos Lelis
;
Athanasios Papakyriakou
;
John Liddle
;
Petros Giastas
, et al.
소스
Proc Natl Acad Sci U S A
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7 .
Discovery of GSK251: A Highly Potent, Highly Selective, Orally Bioavailable Inhibitor of PI3Kδ with a Novel Binding Mode
저자
by
Sebastien Andre Campos
;
Sorif Uddin
;
Daniel Thomas
;
Paul Rowland
;
Birgit Duempelfeld
, et al.
소스
Journal of medicinal chemistry
. 64(18)
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7 .
Reducing False Positives through the Application of Fluorescence Lifetime Technology: A Comparative Study Using TYK2 Kinase as a Model System
저자
by
Peter D. Craggs
;
Faith Mazani
;
Gabriella Clarke
;
Carl Haslam
;
Bhumika Karamshi
, et al.
소스
SLAS discovery : advancing life sciences RD
. 26(5)
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7 . Academic Journal
Optimization ofNovel Indazoles as Highly Potent andSelective Inhibitors of Phosphoinositide 3-Kinase δ forthe Treatment of Respiratory Disease.
저자
by
Kenneth Down
;
Augustin Amour
;
Ian R. Baldwin
;
AnthonyW. J. Cooper
;
Angela M. Deakin
, et al.
소스
Journal of Medicinal Chemistry
. Sep2015, Vol. 58 Issue 18, p7381-7399. 19p.
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7 .
Targeting the Regulatory Site of ER Aminopeptidase 1 Leads to the Discovery of a Natural Product Modulator of Antigen Presentation
저자
by
Jonathan D Lea
;
Robert J. Young
;
Duncan S. Holmes
;
Christopher P. Tinworth
;
Jonathan P. Hutchinson
, et al.
소스
Journal of medicinal chemistry
. 63(6)
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7 .
Design and Development of a Macrocyclic Series Targeting Phosphoinositide 3-Kinase δ
저자
by
Máire A. Convery
;
Daniel Thomas
;
Chris D. Edwards
;
Craig Jamieson
;
James E. Rowedder
, et al.
소스
ACS Med Chem Lett
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7 .
Isoxazolopyrimidine-Based Inhibitors of Plasmodium falciparum Dihydroorotate Dehydrogenase with Antimalarial Activity
저자
by
Margaret A. Phillips
;
David M. Shackleford
;
Jayan T. Joseph
;
Susan A. Charman
;
Jeremy N. Burrows
, et al.
소스
'ACS Omega ', vol: 3, pages: 9227-9240 (2018)
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