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1 . Academic Journal
Activity-Based Protein Profiling of RHBDL4 Reveals Proteolysis of the Enzyme and a Distinct Inhibitor Profile.
저자
by
Davies, Cassondra C.
;
Hu, Ren-Ming
;
Kamitsuka, Paul J.
;
Morais, Gabriel N.
;
de Gonzalez, Regina Stasser
, et al.
소스
ACS Chemical Biology; 8/16/2024, Vol. 19 Issue 8, p1674-1682, 9p
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7 . Academic Journal
Development of succinimide-based inhibitors for the mitochondrial rhomboid protease PARL
저자
by
Parsons, William H.
;
Rutland, Nicholas T.
;
Crainic, Jennifer A.
;
Cardozo, Joaquin M.
;
Chow, Alyssa S.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 October 2021 49
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7 . Academic Journal
Discovery of Potent and Selective Inhibitors against Protein-Derived Electrophilic Cofactors.
저자
by
Wang, Xie
;
Lin, Zongtao
;
Bustin, Katelyn A.
;
McKnight, Nate R.
;
Parsons, William H.
, et al.
소스
Journal of the American Chemical Society; 3/30/2022, Vol. 144 Issue 12, p5377-5388, 12p
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7 . Academic Journal
Potent immunosuppressive C32-O-arylethyl ether derivatives of ascomycin with reduced toxicity
저자
by
Armstrong, Helen M.
;
Wong, Frederick
;
Holmes, Mark A.
;
Sinclair, Peter J.
;
Goulet, Mark T.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1999 9(14):2089-2094
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7 . Academic Journal
C32-O-phenalkyl ether derivatives of the immunosuppressant ascomycin: a tether length study
저자
by
Goulet, Mark T.
;
Sinclair, Peter J.
;
Wong, Frederick
;
Staruch, Mary Jo
;
Dumont, Francis J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1999 9(14):2085-2088
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7 . Periodical
Activity-Based Hydrazine Probes for Protein Profiling of Electrophilic Functionality in Therapeutic Targets
저자
by
Lin, Zongtao
;
Wang, Xie
;
Bustin, Katelyn A.
;
Shishikura, Kyosuke
;
McKnight, Nate R.
, et al.
소스
ACS Central Science; September 2021, Vol. 7 Issue: 9 p1524-1534, 11p
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7 . Academic Journal
Discovery of vinylcycloalkyl-substituted benzimidazole TRPM8 antagonists effective in the treatment of cold allodynia
저자
by
Calvo, Raul R.
;
Meegalla, Sanath K.
;
Parks, Daniel J.
;
Parsons, William H.
;
Ballentine, Shelley K.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 March 2012 22(5):1903-1907
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7 . Academic Journal
AIG1 and ADTRP are endogenous hydrolases of fatty acid esters of hydroxy fatty acids (FAHFAs) in mice.
저자
by
Ertunc, Meric Erikci
;
Kok, Bernard P.
;
Parsons, William H.
;
Wang, Justin G.
;
Dan Tan
, et al.
소스
Journal of Biological Chemistry
. 5/1/2020, Vol. 295 Issue 18, p5891-5905. 15p.
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7 . Academic Journal
Discovery of a novel class of biphenyl pyrazole sodium channel blockers for treatment of neuropathic pain
저자
by
Tyagarajan, Sriram
;
Chakravarty, Prasun K.
;
Zhou, Bishan
;
Taylor, Brett
;
Eid, Ronsar
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(24):7479-7482
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7 . Academic Journal
Substituted biaryl pyrazoles as sodium channel blockers
저자
by
Tyagarajan, Sriram
;
Chakravarty, Prasun K.
;
Zhou, Bishan
;
Taylor, Brett
;
Fisher, Michael H.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(18):5480-5483
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