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1 . Academic Journal
Discovery of potent, selective, bioavailable phosphodiesterase 2 (PDE2) inhibitors active in an osteoarthritis pain model, Part I: Transformation of selective pyrazolodiazepinone phosphodiesterase 4 (PDE4) inhibitors into selective PDE2 inhibitors
저자
by
Plummer, Mark S.
;
Cornicelli, Joseph
;
Roark, Howard
;
Skalitzky, Donald J.
;
Stankovic, Charles J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 June 2013 23(11):3438-3442
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7 . Academic Journal
Discovery of potent selective bioavailable phosphodiesterase 2 (PDE2) inhibitors active in an osteoarthritis pain model. Part II: Optimization studies and demonstration of in vivo efficacy
저자
by
Plummer, Mark S.
;
Cornicelli, Joseph
;
Roark, Howard
;
Skalitzky, Donald J.
;
Stankovic, Charles J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 June 2013 23(11):3443-3447
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7 . Academic Journal
PF-04859989 as a template for structure-based drug design: Identification of new pyrazole series of irreversible KAT II inhibitors with improved lipophilic efficiency
저자
by
Dounay, Amy B.
;
Anderson, Marie
;
Bechle, Bruce M.
;
Evrard, Edelweiss
;
Gan, Xinmin
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 April 2013 23(7):1961-1966
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7 . Academic Journal
Discovery of PF-06835919: A Potent Inhibitor of Ketohexokinase (KHK) for the Treatment of Metabolic Disorders Driven by the Overconsumption of Fructose.
저자
by
Futatsugi, Kentaro
;
Smith, Aaron C.
;
Tu, Meihua
;
Raymer, Brian
;
Ahn, Kay
, et al.
소스
Journal of Medicinal Chemistry; 11/25/2020, Vol. 63 Issue 22, p13546-13560, 15p
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7 . Periodical
Corrections to Design of Selective, ATP-Competitive Inhibitors of Akt
저자
by
Freeman-Cook, Kevin D.
;
Autry, Christopher
;
Borzillo, Gary
;
Gordon, Deborah
;
Barbacci-Tobin, Elsa
, et al.
소스
Journal of Medicinal Chemistry; 20240101, Issue: Preprints
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7 . Periodical
Identification of a Potent, Highly Selective, and Brain Penetrant Phosphodiesterase 2A Inhibitor Clinical Candidate
저자
by
Helal, Christopher J.
;
Arnold, Eric
;
Boyden, Tracey
;
Chang, Cheng
;
Chappie, Thomas A.
, et al.
소스
Journal of Medicinal Chemistry; 20240101, Issue: Preprints
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7 . Periodical
Azetidine and Piperidine Carbamates as Efficient, Covalent Inhibitors of Monoacylglycerol Lipase
저자
by
Butler, Christopher R.
;
Beck, Elizabeth M.
;
Harris, Anthony
;
Huang, Zhen
;
McAllister, Laura A.
, et al.
소스
Journal of Medicinal Chemistry; 20240101, Issue: Preprints
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7 . Academic Journal
6-Amino-4-(pyrimidin-4-yl)pyridones: Novel glycogen synthase kinase-3β inhibitors
저자
by
Coffman, Karen
;
Brodney, Michael
;
Cook, James
;
Lanyon, Lorraine
;
Pandit, Jayvardhan
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(5):1429-1433
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7 . Academic Journal
Synthesis and structure based optimization of novel Akt inhibitors
저자
by
Lippa, Blaise
;
Pan, Gonghua
;
Corbett, Matthew
;
Li, Chao
;
Kauffman, Goss S.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(11):3359-3363
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7 . Academic Journal
Potent, selective spiropyrrolidine pyrimidinetrione inhibitors of MMP-13
저자
by
Freeman-Cook, Kevin D.
;
Reiter, Lawrence A.
;
Noe, Mark C.
;
Antipas, Amy S.
;
Danley, Dennis E.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2007 17(23):6529-6534
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