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1 . Academic Journal
Lead generation from N-[benzyl(4-phenylbutyl)carbamoyl]amino acid as a novel LPA1 antagonist for the treatment of systemic sclerosis
저자
by
Kobayashi, Yuki
;
Uneuchi, Fumito
;
Naruse, Takumi
;
Matsuda, Daisuke
;
Okumura-Kitajima, Lisa
, et al.
소스
In
European Journal of Medicinal Chemistry
15 November 2023 260
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7 . Academic Journal
Design, synthesis and biological evaluation of novel indole derivatives as gut-selective NaPi2b inhibitors
저자
by
Ushiki, Yasunobu
;
Kawabe, Kenichi
;
Yamamoto-Okada, Kumiko
;
Uneuchi, Fumito
;
Asanuma, Yuta
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 July 2022 66
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7 . Academic Journal
Design, synthesis and biological evaluation of novel pyridine derivatives as gut-selective NaPi2b inhibitors
저자
by
Ushiki, Yasunobu
;
Kawabe, Kenichi
;
Yamamoto-Okada, Kumiko
;
Uneuchi, Fumito
;
Asanuma, Yuta
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 June 2022 65
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7 . Academic Journal
Design, synthesis and biological evaluation of novel 1H-pyrazole-4-carbonyl-4,5,6,7-tetrahydrobenzo [b]thiophene derivatives as gut-selective NaPi2b inhibitors
저자
by
Ushiki, Yasunobu
;
Kawabe, Kenichi
;
Yamamoto-Okada, Kumiko
;
Uneuchi, Fumito
;
Asanuma, Yuta
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 March 2022 59
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7 . Academic Journal
Discovery of a potent, low-absorbable sodium-dependent glucose cotransporter 1 (SGLT1) inhibitor (TP0438836) for the treatment of type 2 diabetes
저자
by
Kuroda, Shoichi
;
Kobashi, Yohei
;
Oi, Takahiro
;
Amada, Hideaki
;
Okumura-Kitajima, Lisa
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2018 28(22):3534-3539
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7 . Academic Journal
Discovery of novel 2-[(4-hydroxy-6-oxo-2,3-dihydro-1H-pyridine-5-carbonyl)amino]acetic acid derivatives as HIF prolyl hydroxylase inhibitors for treatment of renal anemia
저자
by
Hamada, Makoto
;
Takayama, Tetsuo
;
Shibata, Tsuyoshi
;
Hiratate, Akira
;
Takahashi, Masato
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 June 2018 28(10):1725-1730
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7 . Academic Journal
SGL5213, a novel and potent intestinal SGLT1 inhibitor, suppresses intestinal glucose absorption and enhances plasma GLP-1 and GLP-2 secretion in rats.
저자
by
Io, Fusayo
;
Gunji, Emi
;
Koretsune, Hiroko
;
Kato, Koji
;
Sugisaki-Kitano, Mami
, et al.
소스
European Journal of Pharmacology
. Jun2019, Vol. 853, p136-144. 9p.
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7 . Academic Journal
Discovery of potent, low-absorbable sodium-dependent glucose cotransporter 1 (SGLT1) inhibitor SGL5213 for type 2 diabetes treatment.
저자
by
Kuroda, Shoichi
;
Kobashi, Yohei
;
Oi, Takahiro
;
Kawabe, Kenichi
;
Shiozawa, Fumiyasu
, et al.
소스
Bioorganic & Medicinal Chemistry
. Jan2019, Vol. 27 Issue 2, p394-409. 16p.
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7 . Academic Journal
Synthesis and Structure-Activity Relationship of C-Phenyl D-Glucitol (TP0454614) Derivatives as Selective Sodium-Dependent Glucose Cotransporter 1 (SGLT1) Inhibitors
저자
by
Kuroda, Shoichi
;
Kobashi, Yohei
;
Kawamura, Madoka
;
Kawabe, Kenichi
;
Shiozawa, Fumiyasu
, et al.
소스
CHEMICAL & PHARMACEUTICAL BULLETIN
; JUL 2020, 68 7, p635-p652, 18p.
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7 . Academic Journal
(2S,4S)-4-Fluoro-1-{[(2-hydroxy-1,1-dimethylethyl)amino]acetyl}-pyrrolidine-2-carbonitrile monobenzenesulfonate (TS-021) is a selective and reversible dipeptidyl peptidase IV inhibitor
저자
by
Tajima, Atsushi
;
Yamamoto, Koji
;
Kozakai, Akinori
;
Okumura-Kitajima, Lisa
;
Mita, Yasuo
, et al.
소스
European Journal of Pharmacology
. Mar 01, 2011 655(1):99-107
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