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1 . Academic Journal
Discovery of novel, potent and orally available benzoazipinone derivatives that elicit MKLP2-inhibitory phenotypes
저자
by
Jian Huang
;
Ting Zhang
;
Julia Kalashova
;
Jinhua Li
;
Chenglu Yang
, et al.
소스
European Journal of Medicinal Chemistry Reports, Vol 11, Iss , Pp 100145- (2024)
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7 . Academic Journal
The Aurora kinase B relocation blocker LXY18 triggers mitotic catastrophe selectively in malignant cells.
저자
by
Julia Kalashova
;
Chenglu Yang
;
Hongmei Li
;
Yan Long
;
Duo Yu
, et al.
소스
PLoS ONE, Vol 18, Iss 10, p e0293283 (2023)
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Scopus
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7 . Academic Journal
The Effect of Circumscribed Exposure to the Pan-Aurora Kinase Inhibitor VX-680 on Proliferating Euploid Cells
저자
by
Xumei Liu
;
Qiong Shi
;
Namrta Choudhry
;
Ting Zhang
;
Hong Liu
, et al.
소스
International Journal of Molecular Sciences, Vol 23, Iss 20, p 12104 (2022)
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7 . Academic Journal
An Oleanolic Acid Derivative Inhibits Hemagglutinin-Mediated Entry of Influenza A Virus
저자
by
Mengdie Ye
;
Yixian Liao
;
Li Wu
;
Wenbao Qi
;
Namrta Choudhry
, et al.
소스
Viruses, Vol 12, Iss 2, p 225 (2020)
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7 .
Discovery and Optimization of Seven-Membered Lactam-Based Compounds to Phenocopy the Inhibition of the Aurora Kinase B
저자
by
Jian Huang
;
Qiong Shi
;
Namrta Choudhry
;
Hongmei Li
;
Chenglu Yang
, et al.
소스
ACS Medicinal Chemistry Letters
. 13:1091-1098
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7 .
An orally bioavailable 4-phenoxy-quinoline compound as a potent AURKB relocation blocker for cancer treatment
저자
by
Jinhua Li
;
Ting Zhang
;
Qiong Shi
;
Gang Lv
;
Xiaohu Zhou
, et al.
소스
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7 .
In-vitro metabolism of LXY18, an orally available, potent blocker of AURKB relocation in mitosis
저자
by
Jinhua Li
;
Namrta Choudhry
;
Gang Lv
;
Naganna Nimishetti
;
Mallu Chenna Reddy
, et al.
소스
Journal of Pharmaceutical and Biomedical Analysis
. 232:115415
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7 .
Integrating a phenotypic screening with a structural simplification strategy to identify 4-phenoxy-quinoline derivatives to potently disrupt the mitotic localization of Aurora kinase B
저자
by
Gang Lv
;
Qiong Shi
;
Ting Zhang
;
Jinhua Li
;
Yan Long
, et al.
소스
Bioorganic & Medicinal Chemistry
. 80:117173
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7 .
2-Phenoxy-3, 4′-bipyridine derivatives inhibit AURKB-dependent mitotic processes by disrupting its localization
저자
by
Gang Lv
;
Qiong Shi
;
Ting Zhang
;
Jinhua Li
;
Julia Kalashova
, et al.
소스
European Journal of Medicinal Chemistry
. 245:114904
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7 .
Exploiting mechanism-informed phenotypic screening for development of next-generation antimitotic phytochemicals
저자
by
Jing Zhang
;
Dun Yang
;
Namrta Choudhry
;
Thaddeus D. Allen
;
Vidhula Ahire
.
소스
Integrative Cancer Science and Therapeutics
. 8
Open Access (OpenAIRE)
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