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1 . Academic Journal
Structurally-defined deubiquitinase inhibitors provide opportunities to investigate disease mechanisms
저자
by
Wertz, Ingrid E.
;
Murray, Jeremy M.
.
소스
In
Drug Discovery Today: Technologies
April 2019 31:109-123
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4 . Academic Journal
Investigation into the mechanism of λmax shifts and their dependence on pH for the 2-hydrazinopyridine derivatives of two copper amine oxidases
저자
by
Saysell, Colin G.
;
Murray, Jeremy M.
;
Wilmot, Carrie M.
;
Brown, Doreen E.
;
Dooley, David M.
, et al.
소스
In
Journal of Molecular Catalysis. B, Enzymatic
2000 8(1):17-25
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7 . Academic Journal
Identification of GNE-293, a potent and selective PI3Kδ inhibitor: Navigating in vitro genotoxicity while improving potency and selectivity
저자
by
Safina, Brian S.
;
Sweeney, Zachary K.
;
Li, Jun
;
Chan, Bryan K.
;
Bisconte, Angelina
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 September 2013 23(17):4953-4959
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7 . Academic Journal
Structure-based discovery of C-2 substituted imidazo-pyrrolopyridine JAK1 inhibitors with improved selectivity over JAK2
저자
by
Labadie, Sharada
;
Dragovich, Peter S.
;
Barrett, Kathy
;
Blair, Wade S.
;
Bergeron, Philippe
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2012 22(24):7627-7633
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7 . Periodical
Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 2: Improvement of In Vitro Antiproliferation Activity and In Vivo Antitumor Efficacy
저자
by
Dragovich, Peter S.
;
Pillow, Thomas H.
;
Blake, Robert A.
;
Sadowsky, Jack D.
;
Adaligil, Emel
, et al.
소스
Journal of Medicinal Chemistry; March 2021, Vol. 64 Issue: 5 p2576-2607, 32p
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7 . Periodical
Discovery of Small-Molecule Inhibitors of Ubiquitin Specific Protease 7 (USP7) Using Integrated NMR and in Silico Techniques
저자
by
Di Lello, Paola
;
Pastor, Richard
;
Murray, Jeremy M.
;
Blake, Robert A.
;
Cohen, Frederick
, et al.
소스
Journal of Medicinal Chemistry; 20240101, Issue: Preprints
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7 . Academic Journal
Structure-based design of thienobenzoxepin inhibitors of PI3-kinase
저자
by
Staben, Steven T.
;
Siu, Michael
;
Goldsmith, Richard
;
Olivero, Alan G.
;
Do, Steven
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 July 2011 21(13):4054-4058
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7 . Academic Journal
Structure-based optimization of pyrazolo-pyrimidine and -pyridine inhibitors of PI3-kinase
저자
by
Staben, Steven T.
;
Heffron, Timothy P.
;
Sutherlin, Daniel P.
;
Bhat, Seema R.
;
Castanedo, Georgette M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(20):6048-6051
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7 . Academic Journal
Discovery of 2-pyrimidyl-5-amidothiophenes as potent inhibitors for AKT: Synthesis and SAR studies
저자
by
Lin, Xiaodong
;
Murray, Jeremy M.
;
Rico, Alice C.
;
Wang, Michael X.
;
Chu, Daniel T.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2006 16(16):4163-4168
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7 . Academic Journal
Discovery of Small-Molecule Inhibitors of Ubiquitin Specific Protease 7 (USP7) Using Integrated NMR and in Silico Techniques.
저자
by
Di Lello, Paola
;
Pastor, Richard
;
Murray, Jeremy M.
;
Blake, Robert A.
;
Cohen, Frederick
, et al.
소스
Journal of Medicinal Chemistry
. 12/28/2017, Vol. 60 Issue 24, p10056-10070. 15p.
Full Text (ACS)
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