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1 . Academic Journal
A rhein-huprine hybrid protects erythrocyte membrane integrity against Alzheimer’s disease related Aβ(1-42) peptide
저자
by
Zambrano, Pablo
;
Jemiola-Rzeminska, Malgorzata
;
Muñoz-Torrero, Diego
;
Suwalsky, Mario
;
Strzalka, Kazimierz
.
소스
In
Biophysical Chemistry
September 2023 300
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7 . Academic Journal
From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effects
저자
by
Pont, Caterina
;
Ginex, Tiziana
;
Griñán-Ferré, Christian
;
Scheiner, Matthias
;
Mattellone, Alexia
, et al.
소스
In
European Journal of Medicinal Chemistry
5 December 2021 225
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7 . Academic Journal
A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors
저자
by
Pérez-Areales, F. Javier
;
Turcu, Andreea L.
;
Barniol-Xicota, Marta
;
Pont, Caterina
;
Pivetta, Deborah
, et al.
소스
In
European Journal of Medicinal Chemistry
15 October 2019 180:613-626
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7 . Academic Journal
First homology model of Plasmodium falciparum glucose-6-phosphate dehydrogenase: Discovery of selective substrate analog-based inhibitors as novel antimalarial agents
저자
by
Alencar, Nelson
;
Sola, Irene
;
Linares, María
;
Juárez-Jiménez, Jordi
;
Pont, Caterina
, et al.
소스
In
European Journal of Medicinal Chemistry
25 February 2018 146:108-122
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7 . Academic Journal
Synthesis and biological evaluation of N-cyanoalkyl-, N-aminoalkyl-, and N-guanidinoalkyl-substituted 4-aminoquinoline derivatives as potent, selective, brain permeable antitrypanosomal agents
저자
by
Sola, Irene
;
Artigas, Albert
;
Taylor, Martin C.
;
Pérez-Areales, F. Javier
;
Viayna, Elisabet
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 November 2016 24(21):5162-5171
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7 . Academic Journal
Design, synthesis and biological evaluation of N-methyl-N-[(1,2,3-triazol-4-yl)alkyl]propargylamines as novel monoamine oxidase B inhibitors
저자
by
Di Pietro, Ornella
;
Alencar, Nelson
;
Esteban, Gerard
;
Viayna, Elisabet
;
Szałaj, Natalia
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 October 2016 24(20):4835-4854
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7 . Academic Journal
A fast and specific method to screen for intracellular amyloid inhibitors using bacterial model systems
저자
by
Navarro, Susanna
;
Carija, Anita
;
Muñoz-Torrero, Diego
;
Ventura, Salvador
.
소스
In
European Journal of Medicinal Chemistry
4 October 2016 121:785-792
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6 . Academic Journal
Multicomponent reaction-based synthesis and biological evaluation of tricyclic heterofused quinolines with multi-trypanosomatid activity
저자
by
Di Pietro, Ornella
;
Vicente-García, Esther
;
Taylor, Martin C.
;
Berenguer, Diana
;
Viayna, Elisabet
, et al.
소스
In
European Journal of Medicinal Chemistry
13 November 2015 105:120-137
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7 . Academic Journal
Synthesis, biological profiling and mechanistic studies of 4-aminoquinoline-based heterodimeric compounds with dual trypanocidal–antiplasmodial activity
저자
by
Sola, Irene
;
Castellà, Sílvia
;
Viayna, Elisabet
;
Galdeano, Carles
;
Taylor, Martin C.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 August 2015 23(16):5156-5167
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7 . Academic Journal
Shogaol–huprine hybrids: Dual antioxidant and anticholinesterase agents with β-amyloid and tau anti-aggregating properties
저자
by
Pérez-Areales, F. Javier
;
Di Pietro, Ornella
;
Espargaró, Alba
;
Vallverdú-Queralt, Anna
;
Galdeano, Carles
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 October 2014 22(19):5298-5307
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