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1 . Academic Journal
Development of potent and selective ULK1/2 inhibitors based on 7-azaindole scaffold with favorable in vivo properties
저자
by
Morozova, Alisa
;
Chan, Sean Chin
;
Bayle, Simon
;
Sun, Luxin
;
Grassie, Dylan
, et al.
소스
In
European Journal of Medicinal Chemistry
15 February 2024 266
Full Text (ScienceDirect)
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7 . Academic Journal
Differential network analysis of ROS1 inhibitors reveals lorlatinib polypharmacology through co-targeting PYK2
저자
by
Liao, Yi
;
Remsing Rix, Lily L.
;
Li, Xueli
;
Fang, Bin
;
Izumi, Victoria
, et al.
소스
In
Cell Chemical Biology
15 February 2024 31(2):284-297
Full Text (ScienceDirect)
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7 . Academic Journal
The reversible inhibitor SR-4835 binds Cdk12/cyclin K in a noncanonical G-loop conformation
저자
by
Schmitz, Maximilian
;
Kaltheuner, Ines H.
;
Anand, Kanchan
;
Düster, Robert
;
Moecking, Jonas
, et al.
소스
In
Journal of Biological Chemistry
January 2024 300(1)
Full Text (ScienceDirect)
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7 . Academic Journal
The dual PI3Kδ/CK1ε inhibitor umbralisib exhibits unique immunomodulatory effects on CLL T cells
저자
by
Maharaj, Kamira
;
Powers, John J.
;
Achille, Alex
;
Mediavilla-Varela, Melanie
;
Gamal, Wael
, et al.
소스
In
Blood Advances
14 July 2020 4(13):3072-3084
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7 . Academic Journal
Development of dual casein kinase 1δ/1ε (CK1δ/ε) inhibitors for treatment of breast cancer
저자
by
Monastyrskyi, Andrii
;
Nilchan, Napon
;
Quereda, Victor
;
Noguchi, Yoshihiko
;
Ruiz, Claudia
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 February 2018 26(3):590-602
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7 . Academic Journal
Enantio‐ and Diastereoselective (Ipc)
2
BOTf‐Mediated Aldol Reactions of Morpholine Carboxamides.
저자
by
Pedzisa, Lee
;
Monastyrskyi, Andrii
;
Parker, Camille D.
;
Roush, William R.
.
소스
Helvetica Chimica Acta
. Dec2023, Vol. 106 Issue 12, p1-9. 9p.
Scopus
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6 . Academic Journal
Going beyond Binary: Rapid Identification of Protein–Protein Interaction Modulators Using a Multifragment Kinetic Target-Guided Synthesis Approach.
저자
by
Nacheva, Katya
;
Kulkarni, Sameer S.
;
Kassu, Mintesinot
;
Flanigan, David
;
Monastyrskyi, Andrii
, et al.
소스
Journal of Medicinal Chemistry; 4/13/2023, Vol. 66 Issue 7, p5196-5207, 12p
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7 . Periodical
Chemical Proteomics with Novel Fully Functionalized Fragments and Stringent Target Prioritization Identifies the Glutathione-Dependent Isomerase GSTZ1 as a Lung Cancer Target
저자
by
Liao, Yi
;
Chin Chan, Sean
;
Welsh, Eric A.
;
Fang, Bin
;
Sun, Luxin
, et al.
소스
ACS Chemical Biology; February 2023, Vol. 18 Issue: 2 p251-264, 14p
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7 . Academic Journal
Discovery of 2-arylquinazoline derivatives as a new class of ASK1 inhibitors
저자
by
Monastyrskyi, Andrii
;
Bayle, Simon
;
Quereda, Victor
;
Grant, Wayne
;
Cameron, Michael
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 February 2018 28(3):400-404
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7 . Periodical
Design and Synthesis of Orally Bioavailable Piperazine Substituted 4(1H)-Quinolones with Potent Antimalarial Activity: Structure–Activity and Structure–Property Relationship Studies
저자
by
Neelarapu, Raghupathi
;
Maignan, Jordany R.
;
Lichorowic, Cynthia L.
;
Monastyrskyi, Andrii
;
Mutka, Tina S.
, et al.
소스
Journal of Medicinal Chemistry; 20240101, Issue: Preprints
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