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1 . Academic Journal
Improvement in oral bioavailability of 2,4-diaminopyrimidine c-Met inhibitors by incorporation of a 3-amidobenzazepin-2-one group
저자
by
Milkiewicz, Karen L.
;
Aimone, Lisa D.
;
Albom, Mark S.
;
Angeles, Thelma S.
;
Chang, Hong
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 November 2011 19(21):6274-6284
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7 . Academic Journal
Synthesis and structure–activity relationships of 1,2,3,4-tetrahydropyrido[2,3- b]pyrazines as potent and selective inhibitors of the anaplastic lymphoma kinase
저자
by
Milkiewicz, Karen L.
;
Weinberg, Linda R.
;
Albom, Mark S.
;
Angeles, Thelma S.
;
Cheng, Mangeng
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2010 18(12):4351-4362
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7 . Academic Journal
Optimization of a novel kinase inhibitor scaffold for the dual inhibition of JAK2 and FAK kinases
저자
by
Zificsak, Craig A.
;
Gingrich, Diane E.
;
Breslin, Henry J.
;
Dunn, Derek D.
;
Milkiewicz, Karen L.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 January 2012 22(1):133-137
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7 . Academic Journal
2,7-Pyrrolo[2,1- f][1,2,4]triazines as JAK2 inhibitors: Modification of target structure to minimize reactive metabolite formation
저자
by
Weinberg, Linda R.
;
Albom, Mark S.
;
Angeles, Thelma S.
;
Breslin, Henry J.
;
Gingrich, Diane E.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(24):7325-7330
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7 . Academic Journal
Fused bicyclic derivatives of 2,4-diaminopyrimidine as c-Met inhibitors
저자
by
Weinberg, Linda R.
;
Albom, Mark S.
;
Angeles, Thelma S.
;
Husten, Jean
;
Lisko, Joseph G.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 January 2011 21(1):164-167
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7 . Academic Journal
Development of a Novel Process for the Kilogram-Scale Synthesis of Spiro[1H‑pyrido[2,3‑d][1,3]oxazine-4,4′-piperidine]-2-one.
저자
by
Mowrey, Dale R.
;
Reif, James J.
;
Milkiewicz, Karen L.
;
Allwein, Shawn P.
.
소스
Organic Process Research & Development; Sep2018, Vol. 22 Issue 9, p1236-1240, 5p
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6 . Academic Journal
Enhanced pharmacokinetic properties of 1,4-benzodiazepine-2,5-dione antagonists of the HDM2-p53 protein–protein interaction through structure-based drug design
저자
by
Parks, Daniel J.
;
LaFrance, Louis V.
;
Calvo, Raul R.
;
Milkiewicz, Karen L.
;
José Marugán, Juan
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2006 16(12):3310-3314
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7 . Academic Journal
1,4-Benzodiazepine-2,5-diones as small molecule antagonists of the HDM2–p53 interaction: discovery and SAR
저자
by
Parks, Daniel J.
;
LaFrance, Louis V.
;
Calvo, Raul R.
;
Milkiewicz, Karen L.
;
Gupta, Varsha
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2005 15(3):765-770
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7 . Academic Journal
Development of a Process Route to the FAK/ALK Dual Inhibitor TEV-37440.
저자
by
Allwein, Shawn P.
;
Mowrey, Dale R.
;
Petrillo, Daniel E.
;
Reif, James J.
;
Purohit, Vikram C.
, et al.
소스
Organic Process Research & Development; May2017, Vol. 21 Issue 5, p740-747, 8p
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7 . Academic Journal
Plant Process for the Preparation of Cinchona Alkaloid-Based Thiourea Catalysts.
저자
by
Yi Wang
;
Milkiewicz, Karen L.
;
Kaufman, Mildred L.
;
Linli He
;
Landmesser, Nelson G.
, et al.
소스
Organic Process Research & Development; Mar2017, Vol. 21 Issue 3, p408-413, 6p
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