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1 .
Discovery of 2,6-disubstituted pyrazine derivatives as inhibitors of CK2 and PIM kinases
저자
by
Emma L. Cooke
;
Xiaoyun Wu
;
Timothy Pontz
;
Les A. Dakin
;
Michael Howard Block
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 28:1336-1341
Web of Science
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7 .
Structure–Cytotoxicity Relationships of Analogues of N14-Desacetoxytubulysin H
저자
by
Michael Howard Block
;
Jay Harper
;
Fengjiang Wang
;
Lakshmaiah Gingipalli
;
Dorin Toader
, et al.
소스
Journal of Medicinal Chemistry
. 59:10781-10787
Web of Science
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7 .
Discovery of 1-Methyl-1H-imidazole Derivatives as Potent Jak2 Inhibitors
저자
by
Tina Howard
;
Jie Shi
;
Kirsten Bell
;
Jon Read
;
Dennis Huszar
, et al.
소스
Journal of Medicinal Chemistry
. 57:144-158
Web of Science
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7 .
Structure and Property Based Design of Pyrazolo[1,5-a]pyrimidine Inhibitors of CK2 Kinase with Activity in Vivo
저자
by
Larry Bao
;
Jamal Carlos Saeh
;
Emma L. Cooke
;
Christopher R. Denz
;
Claudio Chuaqui
, et al.
소스
ACS Medicinal Chemistry Letters
. 4:800-805
Open Access (OpenAIRE)
Web of Science
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7 .
Discovery of (+)-N-(3-Aminopropyl)-N-[1-(5-benzyl-3-methyl-4-oxo-[1,2]thiazolo[5,4-d]pyrimidin-6-yl)-2-methylpropyl]-4-methylbenzamide (AZD4877), a Kinesin Spindle Protein Inhibitor and Potential Anticancer Agent
저자
by
Ellen Freed
;
Lucienne Ronco
;
Timothy Pontz
;
Patrick Brassil
;
Haiqing Hu
, et al.
소스
Journal of Medicinal Chemistry
. 54:6734-6750
Web of Science
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7 .
Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening
저자
by
Mark Zambrowski
;
Rüdiger Kaspera
;
James E. Dowling
;
Edward J. Hennessy
;
Tao Zhang
, et al.
소스
Journal of medicinal chemistry
. 57(23)
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7 .
Cross coupling reactions of organozinc iodides with solid-supported electrophiles: synthesis of 4-substituted benzoic and 3-substituted (E)- and (Z)-propenoic acids and amides
저자
by
Michael Howard Block
;
Richard F. W. Jackson
;
Leslie J. Oates
.
소스
Organic & Biomolecular Chemistry
. 1:140-144
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5 .
Discovery and Optimization of a Series of Carbazole Ureas as NPY5 Antagonists for the Treatment of Obesity
저자
by
Anthony Ladner
;
Michael R. O’Donovan
;
Scott Boyer
;
Andrew D. Roberts
;
Adrian Pickup
, et al.
소스
Journal of Medicinal Chemistry
. 45:3509-3523
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7 .
Discovery of Disubstituted Imidazo[4,5-b]pyridines and Purines as Potent TrkA Inhibitors
저자
by
Hai-Jun Zhang
;
Paul Lyne
;
Ethan Hoffmann
;
Dingwei Yu
;
Michael Howard Block
, et al.
소스
Open Access (OpenAIRE)
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7 .
Discovery of novel benzylidene-1,3-thiazolidine-2,4-diones as potent and selective inhibitors of the PIM-1, PIM-2, and PIM-3 protein kinases
저자
by
James E. Dowling
;
Michelle Lamb
;
Erika Krasnickas Keeton
;
Alexander Hird
;
Erin Code
, et al.
소스
Bioorganicmedicinal chemistry letters
. 22(14)
Full Text (ScienceDirect)
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