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1 . Academic Journal
SAR study of bicyclo[4.1.0]heptanes as melanin-concentrating hormone receptor R1 antagonists: Taming hERG
저자
by
Su, Jing
;
McKittrick, Brian A.
;
Tang, Haiqun
;
Burnett, Duane A.
;
Clader, John W.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2007 15(16):5369-5385
Full Text (ScienceDirect)
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7 . Academic Journal
Discovery of melanin-concentrating hormone receptor R1 antagonists using high-throughput synthesis
저자
by
Su, Jing
;
McKittrick, Brian A.
;
Tang, Haiqun
;
Czarniecki, Michael
;
Greenlee, William J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2005 13(5):1829-1836
Full Text (ScienceDirect)
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7 . Academic Journal
Iminopyrimidinones: A novel pharmacophore for the development of orally active renin inhibitors
저자
by
McKittrick, Brian A.
;
Caldwell, John P.
;
Bara, Thomas
;
Boykow, George
;
Chintala, Madhu
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 April 2015 25(7):1592-1596
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7 . Academic Journal
Identification of 2-aminooxazole amides as acyl-CoA: Diacylglycerol acyltransferase 1 (DGAT1) inhibitors through scaffold hopping strategy
저자
by
Kim, Hyunjin M.
;
Smith, Michelle D.
;
Kim, Jae-Hun
;
Caplen, Mary Ann
;
Chan, Tin Yau
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2013 23(23):6410-6414
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7 . Academic Journal
Structure based design of iminohydantoin BACE1 inhibitors: Identification of an orally available, centrally active BACE1 inhibitor
저자
by
Cumming, Jared N.
;
Smith, Elizabeth M.
;
Wang, Lingyan
;
Misiaszek, Jeffrey
;
Durkin, James
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 April 2012 22(7):2444-2449
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7 . Academic Journal
SAR studies of C2 ethers of 2H-pyrano[2,3-d]pyrimidine-2,4,7(1H,3H)-triones as nicotinic acid receptor (NAR) agonist
저자
by
Huang, Xianhai
;
Su, Jing
;
Rao, Ashwin U.
;
Tang, Haiqun
;
Zhou, Wei
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 January 2012 22(2):854-858
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7 . Academic Journal
Stereoselective synthesis of C-6 hydroxy tricyclic sulfone as a γ-secretase inhibitor
저자
by
Su, Jing
;
Tang, Haiqun
;
McKittrick, Brian A.
.
소스
In
Tetrahedron Letters
29 June 2011 52(26):3382-3385
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5 . Academic Journal
Synthesis and SAR study of tricyclic sulfones as γ-secretase inhibitors: C-6 and C-8 positions
저자
by
Su, Jing
;
Tang, Haiqun
;
McKittrick, Brian A.
;
Xu, Ruo
;
Clader, John W.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(11):3447-3451
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7 . Academic Journal
T-type calcium channel blockers: spiro-piperidine azetidines and azetidinones—optimization, design and synthesis
저자
by
Smith, Elizabeth M.
;
Sorota, Steve
;
Kim, Hyunjin M.
;
McKittrick, Brian A.
;
Nechuta, Terry L.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 August 2010 20(15):4602-4606
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7 . Academic Journal
Discovery of new SCH 39166 analogs as potent and selective dopamine D 1 receptor antagonists
저자
by
Qiang, Li
;
Sasikumar, T.K.
;
Burnett, Duane A.
;
Su, Jing
;
Tang, Haiqun
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(3):836-840
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