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1 . Academic Journal
Novel Quinazoline Derivatives as Highly Effective A2A Adenosine Receptor Antagonists
저자
by
Amélie Laversin
;
Robin Dufossez
;
Raphaël Bolteau
;
Romain Duroux
;
Séverine Ravez
, et al.
소스
Molecules, Vol 29, Iss 16, p 3847 (2024)
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7 . Academic Journal
Jacalin-Curcumin Complex Sensitizes the Breast Cancer MDA-MB-231 Cell Line
저자
by
Lidiya Petrova
;
Nikolay Gergov
;
Marie Stoup
;
Silvina Zapryanova
;
Els J. M. Van Damme
, et al.
소스
International Journal of Molecular Sciences, Vol 24, Iss 24, p 17399 (2023)
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7 . Academic Journal
A Phosphosite Mutant Approach on LRRK2 Links Phosphorylation and Dephosphorylation to Protective and Deleterious Markers, Respectively
저자
by
Antoine Marchand
;
Alessia Sarchione
;
Panagiotis S. Athanasopoulos
;
Hélène Bauderlique-Le Roy
;
Liesel Goveas
, et al.
소스
Cells, Vol 11, Iss 6, p 1018 (2022)
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7 . Academic Journal
The EGF Domains of MUC4 Oncomucin Mediate HER2 Binding Affinity and Promote Pancreatic Cancer Cell Tumorigenesis
저자
by
Nicolas Stoup
;
Maxime Liberelle
;
Céline Schulz
;
Sumeyye Cavdarli
;
Romain Vasseur
, et al.
소스
Cancers, Vol 13, Iss 22, p 5746 (2021)
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7 .
Discovery of a cryptic site at the interface 2 of TEAD – Towards a new family of YAP/TAZ-TEAD inhibitors
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by
Jean-François Guichou
;
Manon Sturbaut
;
Romain Magnez
;
Marie-Christine Chartier-Harlin
;
Patricia Melnyk
, et al.
소스
European Journal of Medicinal Chemistry
European Journal of Medicinal Chemistry, Elsevier, 2021, 226, pp.113835. ⟨10.1016/j.ejmech.2021.113835⟩
European Journal of Medicinal Chemistry, 2021, 226, pp.113835. ⟨10.1016/j.ejmech.2021.113835⟩
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7 .
Synthesis and SAR Studies of Isoquinoline and Tetrahydroisoquinoline Derivatives as Melatonin Receptor Ligands
저자
by
Maxime Liberelle
;
Philippe Delagrange
;
Amélie Laversin
;
Daniel Henri Caignard
;
Nicolas Lebegue
, et al.
소스
ChemMedChem
. 17(3)
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7 .
High ligand efficiency quinazoline compounds as novel A2A adenosine receptor antagonists
저자
by
Raphaël Bolteau
;
Romain Duroux
;
Amélie Laversin
;
Brandon Vreulz
;
Anna Shiriaeva
, et al.
소스
European Journal of Medicinal Chemistry
. 241:114620
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7 .
Rational design of original fused-cycle selective inhibitors of tryptophan 2,3-dioxygenase
저자
by
Arina Kozlova
;
Benoît Van den Eynde
;
Raphaël Frédérick
;
Simon Klaessens
;
Léopold Thabault
, et al.
소스
Journal of Medicinal Chemistry, (2021)
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7 .
Investigation of chalcogen bioisosteric replacement in a series of heterocyclic inhibitors of tryptophan 2,3-dioxygenase
저자
by
Arina Kozlova
;
Marine Deskeuvre
;
Vincent Stroobant
;
Maxime Liberelle
;
Léopold Thabault
, et al.
소스
European journal of medicinal chemistry
. 227
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7 .
The EGF domains of MUC4 oncomucin interact with ErbB2 and mediate tumorigenic activity of cancer cells represent new potential therapeutic targets
저자
by
Romain Vasseur
;
Romain Magnez
;
N Jonckheere
;
Nicolas Renault
;
Nicolas Stoup
, et al.
소스
The FASEB Journal
. 35
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