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1 . Academic Journal
In vitro and in vivo characterization of a novel, highly potent p53-MDM2 inhibitor
저자
by
Vaupel, Andrea
;
Holzer, Philipp
;
Ferretti, Stephane
;
Guagnano, Vito
;
Kallen, Joerg
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 November 2018 28(20):3404-3408
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7 . Academic Journal
Discovery of a novel class of highly potent inhibitors of the p53–MDM2 interaction by structure-based design starting from a conformational argument
저자
by
Furet, Pascal
;
Masuya, Keiichi
;
Kallen, Joerg
;
Stachyra-Valat, Thérèse
;
Ruetz, Stephan
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 October 2016 26(19):4837-4841
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7 . Academic Journal
Discovery of dihydroisoquinolinone derivatives as novel inhibitors of the p53–MDM2 interaction with a distinct binding mode
저자
by
Gessier, François
;
Kallen, Joerg
;
Jacoby, Edgar
;
Chène, Patrick
;
Stachyra-Valat, Thérèse
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 September 2015 25(17):3621-3625
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7 . Academic Journal
Tetra-substituted imidazoles as a new class of inhibitors of the p53–MDM2 interaction
저자
by
Vaupel, Andrea
;
Bold, Guido
;
De Pover, Alain
;
Stachyra-Valat, Thérèse
;
Hergovich Lisztwan, Joanna
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 May 2014 24(9):2110-2114
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7 . Periodical
Extended Solution-phase Peptide Synthesis Strategy Using Isostearyl-Mixed Anhydride Coupling and a New C-Terminal Silyl Ester-Protecting Group for N-Methylated Cyclic Peptide Production
저자
by
Nagaya, Akihiro
;
Murase, Shota
;
Mimori, Yuji
;
Wakui, Kazuya
;
Yoshino, Madoka
, et al.
소스
Organic Process Research & Development; September 2021, Vol. 25 Issue: 9 p2029-2038, 10p
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7 . Academic Journal
Isostearyl Mixed Anhydrides for the Preparation of N‑Methylated Peptides Using C‑Terminally Unprotected N‑Methylamino Acids.
저자
by
Kurasaki, Haruaki
;
Nagaya, Akihiro
;
Kobayashi, Yutaka
;
Matsuda, Ayumu
;
Matsumoto, Masatoshi
, et al.
소스
Organic Letters; 10/16/2020, Vol. 22 Issue 20, p8039-8043, 5p
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7 . Academic Journal
The central valine concept provides an entry in a new class of non peptide inhibitors of the p53–MDM2 interaction
저자
by
Furet, Pascal
;
Chène, Patrick
;
De Pover, Alain
;
Valat, Thérèse Stachyra
;
Lisztwan, Joanna Hergovich
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 May 2012 22(10):3498-3502
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7 . Academic Journal
New pyrazolo[1,5a]pyrimidines as orally active inhibitors of Lck
저자
by
Gommermann, Nina
;
Buehlmayer, Peter
;
von Matt, Anette
;
Breitenstein, Werner
;
Masuya, Keiichi
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 June 2010 20(12):3628-3631
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7 . Academic Journal
Structural States of Hdm2 and HdmX: X‐ray Elucidation of Adaptations and Binding Interactions for Different Chemical Compound Classes.
저자
by
Kallen, Joerg
;
Izaac, Aude
;
Chau, Suzanne
;
Wirth, Emmanuelle
;
Schoepfer, Joseph
, et al.
소스
ChemMedChem; 7/17/2019, Vol. 14 Issue 14, p1305-1314, 10p
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7 . Academic Journal
Overcoming hERG issues for brain-penetrating cathepsin S inhibitors: 2-Cyanopyrimidines. Part 2
저자
by
Irie, Osamu
;
Kosaka, Takatoshi
;
Kishida, Masashi
;
Sakaki, Junichi
;
Masuya, Keiichi
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(19):5280-5284
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