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1 . Academic Journal
Discovery of a fragment hit compound targeting D-Ala:D-Ala ligase of bacterial peptidoglycan biosynthesis
저자
by
Matic Proj
;
Martina Hrast
;
Gregor Bajc
;
Rok Frlan
;
Anže Meden
, et al.
소스
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1, Pp 387-397 (2023)
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7 . Academic Journal
Inhibition of MurA Enzyme from Escherichia coli by Flavonoids and Their Synthetic Analogues
저자
by
Rok Frlan
;
Martina Hrast
;
Stanislav Gobec
.
소스
ACS Omega, Vol 8, Iss 36, Pp 33006-33016 (2023)
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5 . Academic Journal
The Synthesis of (2R)-Aziridine-2-carboxylic Acid Containing Dipeptides
저자
by
Samo Kuzmič
;
Martina Hrast
;
Rok Frlan
.
소스
Acta Chimica Slovenica, Vol 69, Iss 2, Pp 261-270 (2022)
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5 . Academic Journal
Exploring Alternative Pathways to Target Bacterial Type II Topoisomerases Using NBTI Antibacterials: Beyond Halogen-Bonding Interactions
저자
by
Maja Kokot
;
Doroteja Novak
;
Irena Zdovc
;
Marko Anderluh
;
Martina Hrast
, et al.
소스
Antibiotics, Vol 12, Iss 5, p 930 (2023)
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7 . Academic Journal
Potent DNA gyrase inhibitors bind asymmetrically to their target using symmetrical bifurcated halogen bonds
저자
by
Anja Kolarič
;
Thomas Germe
;
Martina Hrast
;
Clare E. M. Stevenson
;
David M. Lawson
, et al.
소스
Nature Communications, Vol 12, Iss 1, Pp 1-13 (2021)
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7 . Academic Journal
Design and Preparation of Antimicrobial Agents
저자
by
Martina Hrast
.
소스
Antibiotics, Vol 11, Iss 12, p 1778 (2022)
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3 . Academic Journal
Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors
저자
by
Péter Ábrányi-Balogh
;
Aaron Keeley
;
György G. Ferenczy
;
László Petri
;
Tímea Imre
, et al.
소스
Pharmaceuticals, Vol 15, Iss 12, p 1484 (2022)
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7 . Academic Journal
Screening of Big Pharma’s Library against Various in-house Biological Targets
저자
by
Damijan Knez
;
Stanislav Gobec
;
Martina Hrast
.
소스
Molecules, Vol 27, Iss 14, p 4484 (2022)
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5 . Academic Journal
Evaluation of the published kinase inhibitor set to identify multiple inhibitors of bacterial ATP-dependent mur ligases
저자
by
Martina Hrast
;
Kaja Rožman
;
Iza Ogris
;
Veronika Škedelj
;
Delphine Patin
, et al.
소스
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 34, Iss 1, Pp 1010-1017 (2019)
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7 . Academic Journal
Inhibition of MurA Enzyme from Escherichia coli and Staphylococcus aureus by Diterpenes from Lepechinia meyenii and Their Synthetic Analogs
저자
by
Macarena Funes Chabán
;
Martina Hrast
;
Rok Frlan
;
Dafni G. Graikioti
;
Constantinos M. Athanassopoulos
, et al.
소스
Antibiotics, Vol 10, Iss 12, p 1535 (2021)
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