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1 .
Macrocyclic Retinoic Acid Receptor-Related Orphan Receptor C2 Inverse Agonists
저자
by
Mark E. Schnute
;
John I. Trujillo
;
Katherine L. Lee
;
Ray Unwalla
;
Felix F. Vajdos
, et al.
소스
ACS Medicinal Chemistry Letters
. 14:191-198
Web of Science
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7 .
Aminopyrazole Carboxamide Bruton's Tyrosine Kinase Inhibitors. Irreversible to Reversible Covalent Reactive Group Tuning
저자
by
Brian Juba
;
Robert Hughes
;
Mihir D. Parikh
;
Erin McCarthy
;
John I. Trujillo
, et al.
소스
ACS medicinal chemistry letters
. 10(1)
Open Access (OpenAIRE)
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7 .
Discovery of 3-Cyano- N-(3-(1-isobutyrylpiperidin-4-yl)-1-methyl-4-(trifluoromethyl)-1 H-pyrrolo[2,3- b]pyridin-5-yl)benzamide: A Potent, Selective, and Orally Bioavailable Retinoic Acid Receptor-Related Orphan Receptor C2 Inverse Agonist
저자
by
Martin Hegen
;
David C. Wood
;
Patrik Rhönnstad
;
Felix Vajdos
;
Atli Thorarensen
, et al.
소스
Journal of medicinal chemistry
. 61(23)
Open Access (OpenAIRE)
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7 .
Discovery of N-(4-Fluoro-3-methoxybenzyl)-6-(2-(((2S,5R)-5-(hydroxymethyl)-1,4-dioxan-2-yl)methyl)-2H-tetrazol-5-yl)-2-methylpyrimidine-4-carboxamide. A Highly Selective and Orally Bioavailable Matrix Metalloproteinase-13 Inhibitor for the Potential Treatment of Osteoarthritis
저자
by
Michael David Rogers
;
Jeffery N. Carroll
;
Mark A. Massa
;
Jeffrey Hitchcock
;
Peter G. Ruminski
, et al.
소스
Journal of Medicinal Chemistry
. 59:313-327
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7 .
Discovery of a Potent and Selective Sphingosine Kinase 1 Inhibitor through the Molecular Combination of Chemotype-Distinct Screening Hits
저자
by
Maureen K. Highkin
;
Matthew D. McReynolds
;
Matthew J. Saabye
;
John W. Rains
;
Kaliapan Iyanar
, et al.
소스
Journal of medicinal chemistry
. 60(6)
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7 .
Modeling the Clinical Phenotype of BTK Inhibition in the Mature Murine Immune System
저자
by
Cheryl Nickerson-Nutter
;
Dean Messing
;
Nilufer P. Seth
;
Sean Keegan
;
John Douhan
, et al.
소스
The Journal of Immunology
. 193:185-197
Open Access (OpenAIRE)
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7 .
A roadmap to evaluate the proteome-wide selectivity of covalent kinase inhibitors
저자
by
John Charles Kath
;
Theodore O. Johnson
;
Landon R. Whitby
;
Benjamin F. Cravatt
;
Baoxian Wei
, et al.
소스
Nature chemical biology
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7 .
Selective Inhibition of BTK Prevents Murine Lupus and Antibody-Mediated Glomerulonephritis
저자
by
Bruce L. Homer
;
Shashi K. Ramaiah
;
Sean Keegan
;
Cheryl Nickerson-Nutter
;
Joy S. Miyashiro
, et al.
소스
The Journal of Immunology
. 191:4540-4550
Open Access (OpenAIRE)
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7 .
Modulation of cellular S1P levels with a novel, potent and specific inhibitor of sphingosine kinase-1
저자
by
Michelle Kraus
;
Jay M. Wendling
;
Olga V. Nemirovskiy
;
John W. Rains
;
Vincent Peterkin
, et al.
소스
Biochemical Journal
. 444:79-88
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7 .
Structure analysis reveals the flexibility of the ADAMTS-5 active site
저자
by
Huey-Sheng Shieh
;
Grace E. Munie
;
Nicole Caspers
;
Alfredo G. Tomasselli
;
James R. Kiefer
, et al.
소스
Protein Science
. 20:735-744
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