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1 .
SAR inspired by aldehyde oxidase (AO) metabolism: Discovery of novel, CNS penetrant tricyclic M4 PAMs
저자
by
Changho Han
;
J. Scott Daniels
;
Alice L. Rodriguez
;
Colleen M. Niswender
;
Alison R. Gregro
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 29:2224-2228
Open Access (OpenAIRE)
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7 .
Cognitive enhancement and antipsychotic-like activity following repeated dosing with the selective M4 PAM VU0467154
저자
by
Nicholas J. Brandon
;
Mark E. Duggan
;
Colleen M. Niswender
;
Jacob Ball
;
Barak W. Gunter
, et al.
소스
Neuropharmacology
. 128:492-502
Open Access (OpenAIRE)
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7 . Academic Journal
Covalent Modifiers: An Orthogonal Approach to Drug Design.
저자
by
Michele H. Potashman
;
Mark E. Duggan
.
소스
Journal of Medicinal Chemistry
. Mar2009, Vol. 52 Issue 5, p1231-1246. 16p.
Full Text (ACS)
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4 .
Challenges in the development of an M 4 PAM preclinical candidate: The discovery, SAR, and in vivo characterization of a series of 3-aminoazetidine-derived amides
저자
by
Meredith J. Noetzel
;
Colleen M. Niswender
;
Jeanette L. Bertron
;
P. Jeffrey Conn
;
Alice L. Rodriguez
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 27:2990-2995
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7 .
Optimization of M 4 positive allosteric modulators (PAMs): The discovery of VU0476406, a non-human primate in vivo tool compound for translational pharmacology
저자
by
Changho Han
;
Eileen M. Engelberg
;
Michael R. Wood
;
Nicholas J. Brandon
;
Frank W. Byers
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 27:2296-2301
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7 .
Challenges in the development of an M 4 PAM in vivo tool compound: The discovery of VU0467154 and unexpected DMPK profiles of close analogs
저자
by
Michael R. Wood
;
Mark E. Duggan
;
Sichen Chang
;
Nicholas J. Brandon
;
Hyekyung P. Cho
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 27:171-175
Open Access (OpenAIRE)
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7 .
Discovery of VU0467485/AZ13713945: An M4 PAM Evaluated as a Preclinical Candidate for the Treatment of Schizophrenia
저자
by
Mark E. Duggan
;
Michael W. Wood
;
Michael R. Wood
;
Craig W. Lindsley
;
Vincent B. Luscombe
, et al.
소스
ACS Medicinal Chemistry Letters
. 8:233-238
Open Access (OpenAIRE)
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7 .
Toward β-Secretase-1 Inhibitors with Improved Isoform Selectivity
저자
by
Karin Kaspersson
;
Ian Gurrell
;
Elisabeth Bäck
;
Samantha Budd Haeberlein
;
Karin Kolmodin
, et al.
소스
Journal of medicinal chemistry
. 61(8)
Scopus
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7 .
Selective Activation of M4 Muscarinic Acetylcholine Receptors Reverses MK-801-Induced Behavioral Impairments and Enhances Associative Learning in Rodents
저자
by
Colleen M. Niswender
;
Carrie K. Jones
;
Michael R. Wood
;
Craig W. Lindsley
;
Frank W. Byers
, et al.
소스
ACS Chemical Neuroscience
Open Access (OpenAIRE)
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7 .
Corrigendum to 'Challenges in the development of an M4 PAM preclinical candidate: The discovery, SAR, and biological characterization of a series of azetidine-derived tertiary amides' [Bioorg. Med. Chem. Lett. 27(23) (2017) 5179–5184]
저자
by
Mark E. Duggan
;
Frank W. Byers
;
Darren W. Engers
;
Craig W. Lindsley
;
Colleen M. Niswender
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 28:3014
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