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1 . Academic Journal
757 M9657, a novel tumor-targeted conditional anti-CD137 agonist displays MSLN-dependent anti-tumor immunity
저자
by
Jacques Moisan
;
Chunxiao Xu
;
Amit Deshpande
;
Joern-Peter Halle
;
Neil Brewis
, et al.
소스
Journal for ImmunoTherapy of Cancer, Vol 9, Iss Suppl 2 (2021)
Open Access (DOAJ)
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7 .
757 M9657, a novel tumor-targeted conditional anti-CD137 agonist displays MSLN-dependent anti-tumor immunity
저자
by
Amit Deshpande
;
Barroq Safi
;
Martina Hubensack
;
Lindsay Webb
;
Rene Schweickhardt
, et al.
소스
Journal for ImmunoTherapy of Cancer, Vol 9, Iss Suppl 2 (2021)
Open Access (OpenAIRE)
Scopus
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7 .
Discovery and Optimization of a Novel Series of Highly Selective JAK1 Kinase Inhibitors
저자
by
Haixia Wang
;
Marat Alimzhanov
;
Paul Lyne
;
Jason Grant Kettle
;
Jie Shi
, et al.
소스
Journal of Medicinal Chemistry
. 61:5235-5244
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7 . Academic Journal
Discovery of 5-Chloro-N2-[(1S)-1-(5-fluoropyrimidin-2-yl)ethyl]-N4-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine (AZD1480) as a Novel Inhibitor of the Jak/Stat Pathway.
저자
by
Stephanos Ioannidis
;
Michelle L. Lamb
;
Tao Wang
;
Lynsie Almeida
;
Michael H. Block
, et al.
소스
Journal of Medicinal Chemistry
. Jan2011, Vol. 54 Issue 1, p262-276. 15p.
Full Text (ACS)
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7 .
Abstract 964: Induction of immunogenic cell death and interferon signaling by carboplatin and the ATR inhibitor M6620 may contribute to anti-tumor activity of M6620-carboplatin-avelumab triplet combination in MC38 tumor model
저자
by
Andree Blaukat
;
Marat Alimzhanov
;
Frank Zenke
;
Christiane Amendt
;
Patricia Soulard
, et al.
소스
Cancer Research
. 80:964-964
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7 .
Potent and Selective CK2 Kinase Inhibitors with Effects on Wnt Pathway Signaling in Vivo
저자
by
Emma Jenkins
;
Larry Bao
;
Christopher R. Denz
;
Andrew D. Ferguson
;
Geoff Holdgate
, et al.
소스
ACS Medicinal Chemistry Letters
. 7:300-305
Open Access (OpenAIRE)
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7 .
Identification of azabenzimidazoles as potent JAK1 selective inhibitors
저자
by
Jon Read
;
Haixia Wang
;
Dennis Huszar
;
Sameer Kawatkar
;
Kelly Goodwin
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 26:60-67
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7 .
Abstract 2269: ATR inhibitor M6620 enhances anti-tumor efficacy of the combination of the anti-PD-L1 antibody avelumab with platinum-based chemotherapy
저자
by
Marat Alimzhanov
;
Patricia Soulard
;
Astrid Zimmermann
;
Andreas Schroeder
;
Keyvan Tadjalli Mehr
, et al.
소스
Cancer Research
. 79:2269-2269
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7 .
Discovery of 1-Methyl-1H-imidazole Derivatives as Potent Jak2 Inhibitors
저자
by
Tina Howard
;
Jie Shi
;
Kirsten Bell
;
Jon Read
;
Dennis Huszar
, et al.
소스
Journal of Medicinal Chemistry
. 57:144-158
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7 .
Structure and Property Based Design of Pyrazolo[1,5-a]pyrimidine Inhibitors of CK2 Kinase with Activity in Vivo
저자
by
Larry Bao
;
Jamal Carlos Saeh
;
Emma L. Cooke
;
Christopher R. Denz
;
Claudio Chuaqui
, et al.
소스
ACS Medicinal Chemistry Letters
. 4:800-805
Open Access (OpenAIRE)
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