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1 . Academic Journal
A phase 1b/2a multicenter study of the safety and preliminary pharmacodynamic effects of selective muscarinic M1 receptor agonist HTL0018318 in patients with mild‐to‐moderate Alzheimer's disease
저자
by
Pradeep J. Nathan
;
S. Babli Millais
;
Alex Godwood
;
Odile Dewit
;
David M. Cross
, et al.
소스
Alzheimer’s & Dementia: Translational Research & Clinical Interventions, Vol 8, Iss 1, Pp n/a-n/a (2022)
Open Access (Wiley)
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Web of Science
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7 .
From structure to clinic: design of a muscarinic M1 receptor agonist with the potential to treat Alzheimer’s disease
저자
by
Andrew B. Tobin
;
Gerard R. Dawson
;
Patrick M. Sexton
;
Nathan Robertson
;
Sophie J. Bradley
, et al.
소스
Open Access (OpenAIRE)
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7 .
Safety, pharmacokinetics and pharmacodynamics of HTL0009936, a selective muscarinic M-1-acetylcholine receptor agonist: A randomized cross-over trial
저자
by
Tim Tasker
;
Charlotte Bakker
;
Giles A. Brown
;
Alastair J. H. Brown
;
Geert Jan Groeneveld
, et al.
소스
British Journal of Clinical Pharmacology, 87(11), 4439-4449. Wiley
British Journal of Clinical Pharmacology
British Journal of Clinical Pharmacology, 87(11), 4439-4449. WILEY
Open Access (OpenAIRE)
Scopus
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7 .
Safety, pharmacokinetics and exploratory pro-cognitive effects of HTL0018318, a selective M1 receptor agonist, in healthy younger adult and elderly subjects: a multiple ascending dose study
저자
by
Geert Jan Groeneveld
;
Tim Tasker
;
Malcolm Peter Weir
;
Jan Liptrot
;
Giles A. Brown
, et al.
소스
Alzheimer’s Research & Therapy, Vol 13, Iss 1, Pp 1-19 (2021)
Alzheimer's Research and Therapy, 13(1). BMC
Open Access (OpenAIRE)
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7 .
First-in-man study to investigate safety, pharmacokinetics and exploratory pharmacodynamics of HTL0018318, a novel M-1-receptor partial agonist for the treatment of dementias
저자
by
Thalia F. van der Doef
;
Jan Liptrot
;
Pradeep J. Nathan
;
Geert Jan Groeneveld
;
Fiona H. Marshall
, et al.
소스
British Journal of Clinical Pharmacology, 87(7), 2945-2955. WILEY
Open Access (OpenAIRE)
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7 .
Extra-helical binding site of a glucagon receptor antagonist
저자
by
Robert M. Cooke
;
Nathan Robertson
;
Markus Koglin
;
Harini Krishnamurthy
;
Ali Jazayeri
, et al.
소스
Nature
. 533:274-277
Web of Science
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7 .
Unifying Family A GPCR Theories of Activation
저자
by
Jonathan S. Mason
;
Malcolm Peter Weir
;
Frank E. Blaney
;
Andrea Bortolato
;
Benjamin G. Tehan
.
소스
Pharmacology & Therapeutics
. 143:51-60
Web of Science
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7 .
Identification of a novel allosteric GLP-1R antagonist HTL26119 using structure-based drug design
저자
by
Fiona H. Marshall
;
Juan Carlos Mobarec
;
Susan H. Brown
;
James C. Errey
;
Stephen P. Andrews
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 29:126611
Web of Science
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7 .
Monoclonal anti-β1-adrenergic receptor antibodies activate G protein signaling in the absence of β-arrestin recruitment
저자
by
Andrei Zhukov
;
Ali Jazayeri
;
Malcolm Peter Weir
;
G. Cseke
;
Jahnavi Pandya-Pathak
, et al.
소스
mAbs
. 6:246-261
Open Access (OpenAIRE)
Web of Science
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7 .
Structure of class B GPCR corticotropin-releasing factor receptor 1
저자
by
Ali Jazayeri
;
Andrea Bortolato
;
Andrew S. Doré
;
Robert M. Cooke
;
Fiona H. Marshall
, et al.
소스
Nature
. 499:438-443
Web of Science
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